Mitogen-activated protein kinase 1
Kinase structure
Kinase:MAPK1 (Erk2)
Family:MAPK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1495
PDB:6DMG
sc-PDB:
KIDFamMap:Search
Release date:2018-12-19
PubMed: 30457858
Chain:A
(Alternate) Model:A
Click to open a 3D viewer
The orthosteric binding pocket


More entries for 6DMG
6DMGAlternative model: BChain: A
6DMGAlternative model: CChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):59.8° (17.2Å)
G-rich loop rotation:56.4°
Quality Score:9.6
Resolution:2.2 Å
Missing Residues:0
Missing Atoms:4
Ligand binding mode
Waters
Cluster
I2
I3
I5
Ligand
No
No
No
Protein
No
No
Yes

Pocket alignment
Uniprot sequence:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME-TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA
Sequence structure:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME_TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA