Platelet derived growth factor receptor alpha
Kinase structure
Kinase:PDGFRA (PDGFRa)
Family:PDGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1803
PDB:6A32
sc-PDB:
KIDFamMap:Search
Release date:2019-06-19
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:out
αC-helix conformation:in
G-rich loop angle (distance):63.3° (19.1Å)
G-rich loop rotation:42.1°
Quality Score:7.2
Resolution:1.87 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I5
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:RVLGSGAFGKVVEVAVKMLALMSELKIMTHLGLNIVNLLGAYIITEYCFYGDLVNYLHKFLASKNCVHRDLAARNVLLICDFGLA
Sequence structure:RVLGSGAFGKVVEVAVKMLALMSELKIMTHLGLNIVNLLGAYIIIEYCFYGDLVNYLHKFLASKNCVHRDLAARNVLLICDFGLA