Mitogen-activated protein kinase 1
Kinase structure
Kinase:MAPK1 (Erk2)
Family:MAPK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1495
PDB:6Q7S
sc-PDB:
KIDFamMap:Search
Release date:2019-06-26
PubMed: 30878562
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 6Q7S
6Q7SAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):60.6° (18Å)
G-rich loop rotation:80.9°
Quality Score:8
Resolution:1.73 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I2
I3
I5
I8
I10
Ligand
No
No
No
No
No
No
Protein
Yes
No
No
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME-TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA
Sequence structure:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME_TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA