EPH receptor A2
Kinase structure
Kinase:EPHA2 (EphA2)
Family:Eph
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1822
PDB:6HEX
sc-PDB:
KIDFamMap:Search
Release date:2019-08-28
Chain:A
(Alternate) Model:C
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The orthosteric binding pocket


More entries for 6HEX
6HEXAlternative model: AChain: A
6HEXAlternative model: BChain: A


Structural information
DFG conformation:out
αC-helix conformation:in
G-rich loop angle (distance):68.2° (20.4Å)
G-rich loop rotation:82.9°
Quality Score:6.8
Resolution:1.41 Å
Missing Residues:2
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I4
I7
Ligand
No
No
No
Protein
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:KVIGAGEFGEVYKVAIKTLDFLGEAGIMGQFSHNIIRLEGVMIITEYMENGALDKFLREYLANMNYVHRDLAARNILVVSDFGLS
Sequence structure:KVIGAGEFGEVYKVAIKTLDFLGEAGIMGQFSHNI_RLEGVMIITEYMENGALDKFLREYLANMNYVHRDLAARNILVVSDFGL_