Mitogen-activated protein kinase kinase 6
Kinase structure
Kinase:MAP2K6
Family:STE7
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2067
PDB:3ENM
sc-PDB:
KIDFamMap:Search
Release date:2009-03-03
PubMed: 19141286
Chain:A
(Alternate) Model:B
Click to open a 3D viewer
The orthosteric binding pocket


More entries for 3ENM
3ENMAlternative model: AChain: A
3ENMAlternative model: AChain: B
3ENMAlternative model: AChain: C
3ENMAlternative model: AChain: D
3ENMAlternative model: BChain: B
3ENMAlternative model: BChain: C
3ENMAlternative model: BChain: D


Structural information
DFG conformation:out-like
αC-helix conformation:na
G-rich loop angle (distance):106.7° (32.2Å)
G-rich loop rotation:30.6°
Quality Score:3.2
Resolution:2.35 Å
Missing Residues:7
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I8
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:MELGRGAYGVVEKMAVKRIRLLMDLDISMRTVPFTVTFYGAWICMELMD-TSLDKFYKQLHSKLSVIHRDVKPSNVLIMCDFGIS
Sequence structure:_ELGRGAYGVVEK_AVKRIRLL_DLDIS_RTVPFTVTFYGAWIC_EL_D_TSLDKFYKQLHSKLSVIHRDVKPSNVLI_CDFGIS