Homeodomain interacting protein kinase 3
Kinase structure
Kinase:HIPK3
Family:DYRK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:2035
PDB:7O7I
sc-PDB:
KIDFamMap:Search
Release date:2021-11-24
PubMed: 34785661
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):51.2° (15.4Å)
G-rich loop rotation:42.6°
Quality Score:9.6
Resolution:2.5 Å
Missing Residues:0
Missing Atoms:4
Ligand binding mode
Waters
Cluster
I1
I5
I10
Ligand
No
No
No
Protein
Yes
No
Yes

Pocket alignment
Uniprot sequence:DFLGRGTFGQVVKVAIKILQGQIEVSILARLSYNFVRAYECCLVFEMLE-QNLYDFLKQKLKSLGLIHADLKPENIMLVIDFGSA
Sequence structure:DFLGRGTFGQVVKVAIKILQGQIEVSILARLSYNFVRAYECCLVFEMLE_QNLYDFLKQKLKSLGLIHADLKPENIMLVIDFGSA