Transforming growth factor beta receptor II
Kinase structure
Kinase:TGFBR2 (TGFbR2)
Family:STKR
Group:TKL
Species:HUMAN
IUPHAR/BPS ID:1795
PDB:8YGZ
sc-PDB:
KIDFamMap:Search
Release date:2024-03-13
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 8YGZ
8YGZAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):48.9° (14.8Å)
G-rich loop rotation:59.1°
Quality Score:8
Resolution:2.1 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I3
I5
I9
Ligand
No
No
No
Protein
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:TLVGKGRFAEVYKVAVKIFSWKTEKDIFSDINENILQFLTAWLITAFHAKGNLQEYLTRGRPKMPIVHRDLKSSNILVLCDFGLS
Sequence structure:TLVGKGRFAEVYKVAVKIFSWKTEKDIFSDINENILQFLTAWLITAFHAKGNLQEYLTRGRPKMPIVHRDLKSSNILVLCDFGLS