WNK lysine deficient protein kinase 1
Kinase structure
Kinase:WNK1 (Wnk1)
Family:WNK
Group:Other
Species:HUMAN
IUPHAR/BPS ID:2280
PDB:4PWN
sc-PDB:
KIDFamMap:Search
Release date:2014-05-28
PubMed: 24803536
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:out
G-rich loop angle (distance):60.4° (17.2Å)
G-rich loop rotation:14.1°
Quality Score:7.6
Resolution:1.84 Å
Missing Residues:1
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I3
I4
I5
Ligand
No
No
No
Protein
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:IEIGRGSFKTVYKVAWCELRFKEEAEMLKGLQPNIVRFYDSVLVTELMTSGTLKTYLKRHTRTPPIIHRDLKCDNIFIIGDLGLA
Sequence structure:IEIGRGSFKTVYKVAWCEL_FKEEAEMLKGLQPNIVRFYDSVLVTELMTSGTLKTYLKRHTRTPPIIHRDLKCDNIFIIGDLGLA