Mitogen-activated protein kinase 1
Kinase structure
Kinase:MAPK1 (Erk2)
Family:MAPK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1495
PDB:4IZA
sc-PDB:
KIDFamMap:Search
Release date:2013-04-10
PubMed: 23575685
Chain:C
(Alternate) Model:A
Click to open a 3D viewer
The orthosteric binding pocket


More entries for 4IZA
4IZAAlternative model: AChain: A
4IZAAlternative model: BChain: A
4IZAAlternative model: BChain: C


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):61° (18.1Å)
G-rich loop rotation:79.2°
Quality Score:8.2
Resolution:1.93 Å
Missing Residues:0
Missing Atoms:18
Ligand binding mode
Waters
Cluster
I3
I8
I10
Ligand
No
No
No
Protein
Yes
Yes
No

Pocket alignment
Uniprot sequence:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME-TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA
Sequence structure:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME_TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA