Mitogen-activated protein kinase 1
Kinase structure
Kinase:MAPK1 (Erk2)
Family:MAPK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1495
PDB:4IZ7
sc-PDB:
KIDFamMap:Search
Release date:2013-04-10
PubMed: 23575685
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 4IZ7
4IZ7Alternative model: AChain: C
4IZ7Alternative model: BChain: A
4IZ7Alternative model: BChain: C


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):62.9° (18.6Å)
G-rich loop rotation:73.9°
Quality Score:9.6
Resolution:1.8 Å
Missing Residues:0
Missing Atoms:4
Ligand binding mode
Waters
Cluster
I3
I5
Ligand
No
No
Protein
Yes
Yes

Pocket alignment
Uniprot sequence:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME-TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA
Sequence structure:SYIGEGAYGMVCSVAIKKIRTLREIKILLRFRENIIGINDIYIVQDLME_TDLYKLLKTYIHSANVLHRDLKPSNLLLICDFGLA