EPH receptor A3
Kinase structure
Kinase:EPHA3 (EphA3)
Family:Eph
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1823
PDB:2QOI
sc-PDB:
KIDFamMap:Search
Release date:2007-08-21
PubMed: 18547520
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 2QOI
2QOIAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):69.7° (20.4Å)
G-rich loop rotation:64.7°
Quality Score:6.8
Resolution:1.25 Å
Missing Residues:3
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I5
I6
I9
I10
Ligand
No
No
No
No
No
Protein
Yes
Yes
Yes
No
Yes

Pocket alignment
Uniprot sequence:KVVGAGEFGEVCSVAIKTLDFLGEASIMGQFDPNIIRLEGVMIVTEYMENGSLDSFLRKYLSDMGYVHRDLAARNILIVSDFGLS
Sequence structure:KVVGAGEFGEVCSVAIKTLDFLGEASIMGQFDPNIIRLEGVMIVTEYMENGSLDSFLRKYLSDMGYVHRDLAARNILIVSDF___