EPH receptor A3
Kinase structure
Kinase:EPHA3 (EphA3)
Family:Eph
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1823
PDB:2GSF
sc-PDB:
KIDFamMap:Search
Release date:2006-06-13
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):68.8° (20.3Å)
G-rich loop rotation:65.2°
Quality Score:8
Resolution:1.77 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I6
Ligand
No
No
Protein
Yes
Yes

Pocket alignment
Uniprot sequence:KVVGAGEFGEVCSVAIKTLDFLGEASIMGQFDPNIIRLEGVMIVTEYMENGSLDSFLRKYLSDMGYVHRDLAARNILIVSDFGLS
Sequence structure:KVVGAGEFGEVCSVAIKTLDFLGEASIMGQFDPNIIRLEGVMIVTEYMENGSLDSFLRKYLSDMGYVHRDLAARNILIVSDFGLS