EPH receptor A3
Kinase structure
Kinase:EPHA3 (EphA3)
Family:Eph
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1823
PDB:2QOK
sc-PDB:
KIDFamMap:Search
Release date:2007-08-28
PubMed: 18547520
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 2QOK
2QOKAlternative model: BChain: A
2QOKAlternative model: CChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):69.2° (20.3Å)
G-rich loop rotation:65°
Quality Score:8
Resolution:1.2 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I2
I5
I6
I7
I10
I11
Ligand
No
No
No
No
No
No
No
Protein
Yes
Yes
Yes
Yes
No
Yes
Yes

Pocket alignment
Uniprot sequence:KVVGAGEFGEVCSVAIKTLDFLGEASIMGQFDPNIIRLEGVMIVTEYMENGSLDSFLRKYLSDMGYVHRDLAARNILIVSDFGLS
Sequence structure:KVVGAGEFGEVCSVAIKTLDFLGEASIMGQFDPNIIRLEGVMIVTEYMENGSLDSFLRKYLSDMGYVHRDLAARNILIVSDFGLA