Cyclin-dependent kinase 1
Kinase structure
Kinase:CDK1 (CDC2)
Family:CDK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1961
PDB:4YC6
sc-PDB:
KIDFamMap:Search
Release date:2015-05-20
PubMed: 25864384
Chain:C
(Alternate) Model:A
Click to open a 3D viewer
The orthosteric binding pocket


More entries for 4YC6
4YC6Alternative model: AChain: A
4YC6Alternative model: AChain: E
4YC6Alternative model: AChain: G
4YC6Alternative model: BChain: A
4YC6Alternative model: BChain: C
4YC6Alternative model: BChain: E
4YC6Alternative model: BChain: G


Structural information
DFG conformation:in
αC-helix conformation:out
G-rich loop angle (distance):51° (14.8Å)
G-rich loop rotation:52.3°
Quality Score:8
Resolution:2.6 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I3
I5
Ligand
No
No
Protein
Yes
Yes

Pocket alignment
Uniprot sequence:EKIGEGTYGVVYKVAMKKITAIREISLLKELRPNIVSLQDVYLIFEFLS-MDLKKYLDSFCHSRRVLHRDLKPQNLLILADFGLA
Sequence structure:EKIGEGTYGVVYKVAMKKITAIREISLLKELRPNIVSLQDVYLIFEFLS_MDLKKYLDSFCHSRRVLHRDLKPQNLLILADFGLA