Kinase insert domain receptor
Kinase structure
Kinase:KDR
Family:VEGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1813
PDB:1VR2
sc-PDB:
KIDFamMap:Search
Release date:2000-03-15
PubMed: 10368301
Chain:A
Click to open a 3D viewer
The orthosteric binding pocket
Structural information
DFG conformation:out-like
αC-helix conformation:in
G-rich loop angle (distance):63.9° (19Å)
G-rich loop rotation:38.2°
Quality Score:7.2
Resolution:2.4 Å
Missing Residues:3
Missing Atoms:16
Ligand binding mode
Waters
Cluster
I1
I5
I7
Ligand
No
No
No
Protein
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:KPLGRGAFGQVIEVAVKMLALMSELKILIHIGLNVVNLLGAMVIVEFCKFGNLSTYLRSFLASRKCIHRDLAARNILLICDFGLA
Sequence structure:KPLGRGAFGQVIEVAVKMLALMSELKILIHIGLNVVNLLGAMVIVEFCKFGNLSTYLRSFLASRKCIHRDLAARNILLICDF___