Mitogen-activated protein kinase kinase kinase 9
Kinase structure
Kinase:MAP3K9 (MLK1)
Family:MLK
Group:TKL
Species:HUMAN
IUPHAR/BPS ID:2084
PDB:4UY9
sc-PDB:
KIDFamMap:Search
Release date:2015-09-30
PubMed: 26637668
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 4UY9
4UY9Alternative model: AChain: B
4UY9Alternative model: BChain: A
4UY9Alternative model: BChain: B


Structural information
DFG conformation:in
αC-helix conformation:out
G-rich loop angle (distance):52.6° (15.5Å)
G-rich loop rotation:67.2°
Quality Score:9.6
Resolution:2.81 Å
Missing Residues:0
Missing Atoms:4
Ligand binding mode
Waters
Cluster
I4
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:EIIGIGGFGKVYRVAVKAANVRQEAKLFAMLKPNIIALRGVCLVMEFARGGPLNRVLSGDEAIVPIIHRDLKSSNILIITDFGLA
Sequence structure:EIIGIGGFGKVYRVAVKAANVRQEAKLFAMLKPNIIALRGVCLVMEFARGGPLNRVLSGDEAIVPIIHRDLKSSNILIITDFGLA