Transforming growth factor beta receptor II
Kinase structure
Kinase:TGFBR2 (TGFbR2)
Family:STKR
Group:TKL
Species:HUMAN
IUPHAR/BPS ID:1795
PDB:5E8V
sc-PDB:
KIDFamMap:Search
Release date:2016-05-11
PubMed: 27139629
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 5E8V
5E8VAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):48.8° (14.9Å)
G-rich loop rotation:58.9°
Quality Score:8.8
Resolution:1.69 Å
Missing Residues:0
Missing Atoms:12
Ligand binding mode
Waters
Cluster
I1
I3
I5
I8
I9
I11
Ligand
No
No
No
No
No
No
Protein
Yes
No
Yes
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:TLVGKGRFAEVYKVAVKIFSWKTEKDIFSDINENILQFLTAWLITAFHAKGNLQEYLTRGRPKMPIVHRDLKSSNILVLCDFGLS
Sequence structure:TLVGKGRFAEVYKVAVKIFSWKTEKDIFSDINENILQFLTAWLITAFHAKGNLQEYLTRGRPKMPIVHRDLKSSNILVLCDFGLS