EPH receptor A2
Kinase structure
Kinase:EPHA2 (EphA2)
Family:Eph
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1822
PDB:5I9U
sc-PDB:
KIDFamMap:Search
Release date:2016-11-09
PubMed: 27685543
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 5I9U
5I9UAlternative model: AChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):67.7° (20.9Å)
G-rich loop rotation:45.7°
Quality Score:8
Resolution:1.89 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I2
I3
I4
I5
I10
Ligand
No
No
No
No
No
No
Protein
Yes
No
No
Yes
No
Yes

Pocket alignment
Uniprot sequence:KVIGAGEFGEVYKVAIKTLDFLGEAGIMGQFSHNIIRLEGVMIITEYMENGALDKFLREYLANMNYVHRDLAARNILVVSDFGLS
Sequence structure:KVIGAGEFGEVYKVAIKTLDFLGEAGIMGQFSHNIIRLEGVMIITEYMENGALDKFLREYLANMNYVHRDLAARNILVVSDFGLS