Epidermal growth factor receptor
Kinase structure
Kinase:EGFR
Family:EGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1797
PDB:4I21
sc-PDB:
KIDFamMap:Search
Release date:2013-01-16
PubMed: 23273428
Chain:A
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The orthosteric binding pocket


More entries for 4I21
4I21Chain: B


Structural information
DFG conformation:out-like
αC-helix conformation:in
G-rich loop angle (distance):50° (15.3Å)
G-rich loop rotation:18.6°
Quality Score:8
Resolution:3.37 Å
Missing Residues:0
Missing Atoms:0

Pocket alignment
Uniprot sequence:KVLGSGAFGTVYKVAIKELEILDEAYVMASVDPHVCRLLGIQLITQLMPFGCLLDYVREYLEDRRLVHRDLAARNVLVITDFGLA
Sequence structure:KVLGSGAFGTVYKVAIKELEILDEAYVMASVDPHVCRLLGIQLIMQLMPFGCLLDYVREYLEDRRLVHRDLAARNVLVITDFGRA