Epidermal growth factor receptor
Kinase structure
Kinase:EGFR
Family:EGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1797
PDB:4I1Z
sc-PDB:
KIDFamMap:Search
Release date:2013-01-16
PubMed: 23273428
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 4I1Z
4I1ZAlternative model: BChain: A


Structural information
DFG conformation:out-like
αC-helix conformation:in
G-rich loop angle (distance):47.6° (14.6Å)
G-rich loop rotation:30.6°
Quality Score:8
Resolution:3 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I6
Ligand
No
No
Protein
Yes
Yes

Pocket alignment
Uniprot sequence:KVLGSGAFGTVYKVAIKELEILDEAYVMASVDPHVCRLLGIQLITQLMPFGCLLDYVREYLEDRRLVHRDLAARNVLVITDFGLA
Sequence structure:KVLGSGAFGTVYKVAIKELEILDEAYVMASVDPHVCRLLGIQLIMQLMPFGCLLDYVREYLEDRRLVHRDLAARNVLVITDFGRA