PDB-code
Browse kinase entries (page 105 of 282)
First 101 102 103 PreviousLast109 108 107 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | EGFR | EGFR | TK | 6lud | A | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6p1d | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1d | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1d | B | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1d | B | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1d | C | A | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1d | C | B | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1d | D | A | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1d | D | B | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p1l | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6p1l | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6p1l | C | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6p1l | D | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6p8q | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p8q | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p8q | B | A | adenosine monophosphate | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p8q | B | B | adenosine monophosphate | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p8q | C | A | adenosine monophosphate | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p8q | C | B | adenosine monophosphate | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p8q | D | A | adenosine monophosphate | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6p8q | D | B | adenosine monophosphate | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6s89 | A | ~{n}-[3-[6-[4-(4-methylpiperazin-1-yl)phenyl]-4-propan-2-yloxy-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6s8a | A | ~{n}-[3-[6-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-methylpropoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6s9b | A | 3-fluoranyl-~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-5-pyridin-3-yl-benzamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6s9c | A | A | ~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-2-phenyl-pyridine-4-carboxamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6s9c | A | B | ~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-2-phenyl-pyridine-4-carboxamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6s9d | A | 8-oxa-14,21,23,28-tetraazapentacyclo[23.3.1.02,7.014,22.015,20]nonacosa-1(28),2(7),3,5,15,17,19,21,25(29),26-decaen-24-one | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6tfu | A | ~{n}-[3-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6tfu | B | ~{n}-[3-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6tfv | A | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfv | A | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfv | B | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfv | B | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfw | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6tfw | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 6tfy | A | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfy | A | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfy | B | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfy | B | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfz | A | A | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfz | A | B | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfz | B | A | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tfz | B | B | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tg0 | A | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tg0 | A | B | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tg0 | B | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tg0 | B | B | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tg1 | A | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tg1 | A | B | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 6tg1 | B | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | Show | ![]() |


