PDB-code
Browse kinase entries (page 122 of 282)
First 118 119 120 PreviousLast126 125 124 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | FGFR1 | FGFR | TK | 5flf | B | B | - | Human | Show |  |
| FGFR1 | FGFR | TK | 5flf | C | A | - | Human | Show | |
| FGFR1 | FGFR | TK | 5flf | C | B | - | Human | Show | |
| FGFR1 | FGFR | TK | 5flf | D | A | - | Human | Show | |
| FGFR1 | FGFR | TK | 5flf | D | B | - | Human | Show | |
| FGFR1 | FGFR | TK | 5flf | E | A | - | Human | Show | |
| FGFR1 | FGFR | TK | 5flf | E | B | - | Human | Show | |
| FGFR1 | FGFR | TK | 5o49 | A | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5o49 | A | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5o49 | B | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5o49 | B | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5o4a | A | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5o4a | A | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5o4a | B | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5o4a | B | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | Show | |
| FGFR1 | FGFR | TK | 5uq0 | A | A | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | Show | |
| FGFR1 | FGFR | TK | 5uq0 | A | B | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | Show | |
| FGFR1 | FGFR | TK | 5uq0 | B | A | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | Show | |
| FGFR1 | FGFR | TK | 5uq0 | B | B | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | Show | |
| FGFR1 | FGFR | TK | 5ur1 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 5ur1 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 5ur1 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 5ur1 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 5vnd | A | A | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | Show | |
| FGFR1 | FGFR | TK | 5vnd | A | B | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | Show | |
| FGFR1 | FGFR | TK | 5vnd | B | A | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | Show | |
| FGFR1 | FGFR | TK | 5vnd | B | B | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | Show | |
| FGFR1 | FGFR | TK | 5z0s | A | A | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | Show | |
| FGFR1 | FGFR | TK | 5z0s | A | B | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | Show | |
| FGFR1 | FGFR | TK | 5z0s | B | A | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | Show | |
| FGFR1 | FGFR | TK | 5z0s | B | B | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | Show | |
| FGFR1 | FGFR | TK | 5zv2 | A | 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide | Human | Show | | |
| FGFR1 | FGFR | TK | 5zv2 | B | 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide | Human | Show | | |
| FGFR1 | FGFR | TK | 6c18 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c18 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c18 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c18 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c19 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c19 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c19 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c19 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1b | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1b | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1b | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1b | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1c | A | A | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1c | A | B | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1c | B | A | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1c | B | B | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | |
| FGFR1 | FGFR | TK | 6c1o | A | A | n-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamide | Human | Show | |
