Browse kinase entries (page 130 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
GSK3BGSKCMGC1q5kBn-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaHumanShow
GSK3BGSKCMGC1r0eAA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHumanShow
GSK3BGSKCMGC1r0eAB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHumanShow
GSK3BGSKCMGC1r0eBA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHumanShow
GSK3BGSKCMGC1r0eBB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHumanShow
GSK3BGSKCMGC1uv5A6-bromoindirubin-3'-oximeHumanShow
GSK3BGSKCMGC2jldAAruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC2jldABruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC2jldBAruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC2jldBBruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC2o5kA2-(2,4-dichloro-phenyl)-7-hydroxy-1h-benzoimidazole-4-carboxylic acid [2-(4-methanesulfonylamino-phenyl)-ethyl]-amideHumanShow
GSK3BGSKCMGC2ow3Abis-(indole)maleimide pyridinophaneHumanShow
GSK3BGSKCMGC2ow3Bbis-(indole)maleimide pyridinophaneHumanShow
GSK3BGSKCMGC3du8A(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHumanShow
GSK3BGSKCMGC3du8B(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHumanShow
GSK3BGSKCMGC3f7zAA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3f7zAB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3f7zAC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3f7zBA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3f7zBB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3f7zBC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3f88AA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHumanShow
GSK3BGSKCMGC3f88AB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHumanShow
GSK3BGSKCMGC3f88BA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHumanShow
GSK3BGSKCMGC3f88BB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHumanShow
GSK3BGSKCMGC3gb2AA2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3gb2AB2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHumanShow
GSK3BGSKCMGC3i4bAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHumanShow
GSK3BGSKCMGC3i4bBn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHumanShow
GSK3BGSKCMGC3l1sA(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHumanShow
GSK3BGSKCMGC3l1sB(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHumanShow
GSK3BGSKCMGC3m1sAAruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC3m1sABruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC3m1sBAruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC3m1sBBruthenium pyridocarbazoleHumanShow
GSK3BGSKCMGC3pupAruthenium octasporineHumanShow
GSK3BGSKCMGC3pupBruthenium octasporineHumanShow
GSK3BGSKCMGC3q3bA4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHumanShow
GSK3BGSKCMGC3q3bB4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHumanShow
GSK3BGSKCMGC3sayAA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHumanShow
GSK3BGSKCMGC3sayAB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHumanShow
GSK3BGSKCMGC3sayBA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHumanShow
GSK3BGSKCMGC3sayBB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHumanShow
GSK3BGSKCMGC3sd0A3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHumanShow
GSK3BGSKCMGC3sd0B3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHumanShow
GSK3BGSKCMGC3zdiA3,6-diamino-4-(2-chlorophenyl)thieno[2,3-b]pyridine-2,5-dicarbonitrileHumanShow
GSK3BGSKCMGC3zrkAA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHumanShow
GSK3BGSKCMGC3zrkAB2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHumanShow
GSK3BGSKCMGC3zrkAC2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHumanShow
GSK3BGSKCMGC3zrkBA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHumanShow
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