PDB-code
Browse kinase entries (page 131 of 282)
First 127 128 129 PreviousLast135 134 133 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | GSK3B | GSK | CMGC | 3zrk | B | B | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrk | B | C | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrl | A | A | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrl | A | B | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrl | A | C | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrl | B | A | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrl | B | B | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrl | B | C | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrm | A | A | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrm | A | B | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrm | A | C | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrm | B | A | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrm | B | B | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 3zrm | B | C | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4acc | A | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4acc | B | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4acd | A | 3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4acd | B | 3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4acg | A | 2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4acg | B | 2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4ach | A | 3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4ach | B | 3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4afj | A | A | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4afj | A | B | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4afj | A | C | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4afj | B | A | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4afj | B | B | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4afj | B | C | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4b7t | A | (5z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-methyl-2-(propan-2-ylamino)imidazol-4-one | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4dit | A | n-(pyridin-3-yl)-2-(thiophen-3-yl)-3h-imidazo[4,5-b]pyridine-7-carboxamide | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4iq6 | A | 6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amine | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4iq6 | B | 6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amine | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4j1r | A | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4j1r | B | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4j1r | C | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4j1r | D | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() | |
![]() | GSK3B | GSK | CMGC | 4j71 | A | A | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4j71 | A | B | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4j71 | B | A | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4j71 | B | B | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm0 | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm0 | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm3 | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm3 | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm5 | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm5 | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm7 | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4nm7 | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4ptc | A | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | Show | ![]() |
![]() | GSK3B | GSK | CMGC | 4ptc | A | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | Show | ![]() |


