Browse kinase entries (page 132 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
GSK3BGSKCMGC4ptcBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHumanShow
GSK3BGSKCMGC4ptcBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHumanShow
GSK3BGSKCMGC4pteAAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHumanShow
GSK3BGSKCMGC4pteABn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHumanShow
GSK3BGSKCMGC4pteBAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHumanShow
GSK3BGSKCMGC4pteBBn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHumanShow
GSK3BGSKCMGC4ptgAA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHumanShow
GSK3BGSKCMGC4ptgAB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHumanShow
GSK3BGSKCMGC4ptgBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHumanShow
GSK3BGSKCMGC4ptgBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHumanShow
GSK3BGSKCMGC5f94AA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC5f94AB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC5f94BA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC5f94BB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC5f95A2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC5f95B2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC5hlnAchir99021HumanShow
GSK3BGSKCMGC5hlnBchir99021HumanShow
GSK3BGSKCMGC5hlpAA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5hlpAB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5hlpBA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5hlpBB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5k5nA5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHumanShow
GSK3BGSKCMGC5k5nB5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHumanShow
GSK3BGSKCMGC5kpkA(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5kpkB(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5kplAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5kplAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5kplBA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5kplBB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5kpmA(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5kpmB(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5oy4A~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHumanShow
GSK3BGSKCMGC5oy4B~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHumanShow
GSK3BGSKCMGC5t31A(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC5t31B(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC6b8jAAchir99021HumanShow
GSK3BGSKCMGC6b8jABchir99021HumanShow
GSK3BGSKCMGC6gjoA(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHumanShow
GSK3BGSKCMGC6gjoB(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHumanShow
GSK3BGSKCMGC6gn1A~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHumanShow
GSK3BGSKCMGC6gn1B~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHumanShow
GSK3BGSKCMGC6h0uA(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHumanShow
GSK3BGSKCMGC6h0uB(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHumanShow
GSK3BGSKCMGC6hk3AA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6hk3AB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6hk3BA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6hk3BB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6hk4AA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6hk4AB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHumanShow
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