Browse kinase entries (page 133 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
GSK3BGSKCMGC6hk4BA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6hk4BB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6hk7A3-azanyl-~{n}-(2-methoxyethyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHumanShow
GSK3BGSKCMGC6tcuAA5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHumanShow
GSK3BGSKCMGC6tcuAB5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHumanShow
GSK3BGSKCMGC6v6lAA-HumanShow
GSK3BGSKCMGC6v6lAB-HumanShow
GSK3BGSKCMGC6y9rAA~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHumanShow
GSK3BGSKCMGC6y9rAB~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHumanShow
GSK3BGSKCMGC6y9sAA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHumanShow
GSK3BGSKCMGC6y9sAB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHumanShow
GSK3BGSKCMGC6y9sBA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHumanShow
GSK3BGSKCMGC6y9sBB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHumanShow
GSK3BGSKCMGC7b6fAA3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHumanShow
GSK3BGSKCMGC7b6fAB3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHumanShow
GSK3BGSKCMGC7oy5AA~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHumanShow
GSK3BGSKCMGC7oy5AB~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHumanShow
GSK3BGSKCMGC7sxhAA(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHumanShow
GSK3BGSKCMGC7sxhAB(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHumanShow
GSK3BGSKCMGC7sxjAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC7sxjAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHumanShow
GSK3BGSKCMGC7u2zAA(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHumanShow
GSK3BGSKCMGC7u2zAB(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHumanShow
GSK3BGSKCMGC7u31AA5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHumanShow
GSK3BGSKCMGC7u31AB5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHumanShow
GSK3BGSKCMGC7u33AA3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHumanShow
GSK3BGSKCMGC7u33AB3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHumanShow
GSK3BGSKCMGC7u36A(3s)-1-[(2-fluorophenoxy)acetyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHumanShow
GSK3BGSKCMGC7z1fA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
GSK3BGSKCMGC7z1gA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
GSK3BGSKCMGC8auzAA8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHumanShow
GSK3BGSKCMGC8auzAB8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHumanShow
GSK3BGSKCMGC8av1AA2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHumanShow
GSK3BGSKCMGC8av1AB2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHumanShow
GSK3BGSKCMGC8djcAA(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHumanShow
GSK3BGSKCMGC8djcAB(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHumanShow
GSK3BGSKCMGC8djdAA2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC8djdAB2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHumanShow
GSK3BGSKCMGC8djeAA(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHumanShow
GSK3BGSKCMGC8djeAB(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHumanShow
GSK3BGSKCMGC8ff8A2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamideHumanShow
GSK3BGSKCMGC8qjiAn-[4-[5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl]pyridin-2-yl]cyclopropanecarboxamideHumanShow
GUCY2C (HSER)RGCRGC8fx4D-HumanShow
HASPIN (Haspin)HaspinOther2vuwAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther2vuwAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHumanShow
HASPIN (Haspin)HaspinOther2wb8AA-HumanShow
HASPIN (Haspin)HaspinOther2wb8AB-HumanShow
HASPIN (Haspin)HaspinOther3dlzAAadenosine monophosphateHumanShow
HASPIN (Haspin)HaspinOther3dlzABadenosine monophosphateHumanShow
HASPIN (Haspin)HaspinOther3e7vAA3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amineHumanShow
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