Browse kinase entries (page 15 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
ANTXR1 (DNAPK)PIKKAtypical8bhyA-HumanShow
ANTXR1 (DNAPK)PIKKAtypical8ezbCadenosine-5'-triphosphateHumanShow
ATMPIKKAtypical5np0A-HumanShow
ATMPIKKAtypical5np0B-HumanShow
ATMPIKKAtypical5np1A-HumanShow
ATMPIKKAtypical6k9kA-HumanShow
ATMPIKKAtypical6k9lA-HumanShow
ATMPIKKAtypical6k9lB-HumanShow
ATMPIKKAtypical7ni4A8-(1,3-dimethylpyrazol-4-yl)-1-(3-fluoranyl-5-methoxy-pyridin-4-yl)-7-methoxy-3-methyl-imidazo[4,5-c]quinolin-2-oneHumanShow
ATMPIKKAtypical7ni5A2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-oneHumanShow
ATMPIKKAtypical7ni6Aphosphothiophosphoric acid-adenylate esterHumanShow
ATMPIKKAtypical7sicAphosphoaminophosphonic acid-adenylate esterHumanShow
ATMPIKKAtypical7sidAphosphoaminophosphonic acid-adenylate esterHumanShow
ATMPIKKAtypical8oxmBphosphoaminophosphonic acid-adenylate esterHumanShow
ATMPIKKAtypical8oxoBphosphoaminophosphonic acid-adenylate esterHumanShow
ATMPIKKAtypical8oxpAphosphoaminophosphonic acid-adenylate esterHumanShow
ATMPIKKAtypical8oxqAphosphoaminophosphonic acid-adenylate esterHumanShow
ATRPIKKAtypical5yz0A-HumanShow
ATRPIKKAtypical5yz0B-HumanShow
Aurka (AurA)AUROther3d14AA1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouseShow
Aurka (AurA)AUROther3d14AB1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouseShow
Aurka (AurA)AUROther3d15AA1-(3-chlorophenyl)-3-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}ureaMouseShow
Aurka (AurA)AUROther3d2iA1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouseShow
Aurka (AurA)AUROther3d2kA(7-{[2-(2-{[(3-chlorophenyl)carbamoyl]amino}-1,3-thiazol-5-yl)ethyl]amino}-1h-pyrazolo[4,3-d]pyrimidin-1-yl)acetic acidMouseShow
Aurka (AurA)AUROther3dajAn-butyl-3-{[6-(9h-purin-6-ylamino)hexanoyl]amino}benzamideMouseShow
Aurka (AurA)AUROther3dj5A3-({3-[(6-amino-5-bromopyrimidin-4-yl)sulfanyl]propanoyl}amino)-4-methoxy-n-phenylbenzamideMouseShow
Aurka (AurA)AUROther3dj6A4-methoxy-n-phenyl-3-({3-[(1h-pyrrolo[2,3-b]pyridin-5-ylmethyl)sulfanyl]propanoyl}amino)benzamideMouseShow
Aurka (AurA)AUROther3dj7AA1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouseShow
AURKA (AurA)AurOther1mq4Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther1muoAadenosineHumanShow
AURKA (AurA)AurOther1ol5Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther1ol6Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther1ol7Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2bmcA(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2bmcB(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2bmcC(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2bmcD(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2bmcE(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2bmcF(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2c6dAAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther2c6dABphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther2c6eAn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHumanShow
AURKA (AurA)AurOther2c6eBn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHumanShow
AURKA (AurA)AurOther2dwbAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther2j4zA4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHumanShow
AURKA (AurA)AurOther2j4zB4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHumanShow
AURKA (AurA)AurOther2j50An-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther2j50Bn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther2np8An-{3-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]phenyl}cyclopropanecarboxamideHumanShow
AURKA (AurA)AurOther2w1cA4-{[2-(4-{[(4-fluorophenyl)carbonyl]amino}-1h-pyrazol-3-yl)-1h-benzimidazol-6-yl]methyl}morpholin-4-iumHumanShow
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