PDB-code
Browse kinase entries (page 15 of 282)
First 11 12 13 PreviousLast19 18 17 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | ANTXR1 (DNAPK) | PIKK | Atypical | 8bhy | A | - | Human | Show | ![]() | |
![]() | ANTXR1 (DNAPK) | PIKK | Atypical | 8ezb | C | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 5np0 | A | - | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 5np0 | B | - | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 5np1 | A | - | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 6k9k | A | - | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 6k9l | A | - | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 6k9l | B | - | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 7ni4 | A | 8-(1,3-dimethylpyrazol-4-yl)-1-(3-fluoranyl-5-methoxy-pyridin-4-yl)-7-methoxy-3-methyl-imidazo[4,5-c]quinolin-2-one | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 7ni5 | A | 2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 7ni6 | A | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 7sic | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 7sid | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 8oxm | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 8oxo | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 8oxp | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | ATM | PIKK | Atypical | 8oxq | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | ATR | PIKK | Atypical | 5yz0 | A | - | Human | Show | ![]() | |
![]() | ATR | PIKK | Atypical | 5yz0 | B | - | Human | Show | ![]() | |
![]() | Aurka (AurA) | AUR | Other | 3d14 | A | A | 1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]urea | Mouse | Show | ![]() |
![]() | Aurka (AurA) | AUR | Other | 3d14 | A | B | 1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]urea | Mouse | Show | ![]() |
![]() | Aurka (AurA) | AUR | Other | 3d15 | A | A | 1-(3-chlorophenyl)-3-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}urea | Mouse | Show | ![]() |
![]() | Aurka (AurA) | AUR | Other | 3d2i | A | 1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]urea | Mouse | Show | ![]() | |
![]() | Aurka (AurA) | AUR | Other | 3d2k | A | (7-{[2-(2-{[(3-chlorophenyl)carbamoyl]amino}-1,3-thiazol-5-yl)ethyl]amino}-1h-pyrazolo[4,3-d]pyrimidin-1-yl)acetic acid | Mouse | Show | ![]() | |
![]() | Aurka (AurA) | AUR | Other | 3daj | A | n-butyl-3-{[6-(9h-purin-6-ylamino)hexanoyl]amino}benzamide | Mouse | Show | ![]() | |
![]() | Aurka (AurA) | AUR | Other | 3dj5 | A | 3-({3-[(6-amino-5-bromopyrimidin-4-yl)sulfanyl]propanoyl}amino)-4-methoxy-n-phenylbenzamide | Mouse | Show | ![]() | |
![]() | Aurka (AurA) | AUR | Other | 3dj6 | A | 4-methoxy-n-phenyl-3-({3-[(1h-pyrrolo[2,3-b]pyridin-5-ylmethyl)sulfanyl]propanoyl}amino)benzamide | Mouse | Show | ![]() | |
![]() | Aurka (AurA) | AUR | Other | 3dj7 | A | A | 1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]urea | Mouse | Show | ![]() |
![]() | AURKA (AurA) | Aur | Other | 1mq4 | A | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 1muo | A | adenosine | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 1ol5 | A | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 1ol6 | A | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 1ol7 | A | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2bmc | A | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2bmc | B | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2bmc | C | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2bmc | D | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2bmc | E | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2bmc | F | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2c6d | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | AURKA (AurA) | Aur | Other | 2c6d | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | AURKA (AurA) | Aur | Other | 2c6e | A | n-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2c6e | B | n-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2dwb | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2j4z | A | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2j4z | B | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2j50 | A | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2j50 | B | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2np8 | A | n-{3-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]phenyl}cyclopropanecarboxamide | Human | Show | ![]() | |
![]() | AURKA (AurA) | Aur | Other | 2w1c | A | 4-{[2-(4-{[(4-fluorophenyl)carbonyl]amino}-1h-pyrazol-3-yl)-1h-benzimidazol-6-yl]methyl}morpholin-4-ium | Human | Show | ![]() |


