PDB-code
Browse kinase entries (page 17 of 282)
First 13 14 15 PreviousLast21 20 19 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | AURKA (AurA) | Aur | Other | 3unz | B | 4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | Show |  | |
| AURKA (AurA) | Aur | Other | 3uo4 | A | 4-{[4-(biphenyl-2-ylamino)pyrimidin-2-yl]amino}benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uo5 | A | 4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uo6 | A | 4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uo6 | B | 4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uod | A | 4-[(4-{[2-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uoh | A | 4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uoh | B | 4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uoj | A | 4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uoj | B | 4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uok | A | 4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uok | B | 4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uol | A | n~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamine | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3uol | B | n~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamine | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3up2 | A | 4-[(4-{[2-(trifluoromethoxy)phenyl]amino}pyrimidin-2-yl)amino]benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3up7 | A | 2-({2-[(4-carboxyphenyl)amino]pyrimidin-4-yl}amino)benzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3vap | A | 3-(1-{2-[(3-fluoropyridinium-4-yl)amino]-2-oxoethyl}-1h-pyrazol-4-yl)-6-methyl-8-[(3-{[(1r,3r)-3-methylpiperidinium-1-yl]methyl}-1,2-thiazol-5-yl)amino]imidazo[1,2-a]pyrazin-1-ium | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w10 | A | 1-(3-methoxyphenyl)-n-(5-methyl-1h-pyrazol-3-yl)isoquinolin-3-amine | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w16 | A | 4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-one | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w18 | A | 2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w18 | B | 2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w2c | A | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w2c | C | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w2c | E | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 3w2c | G | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4b0g | A | A | 6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridine | Human | Show | |
| AURKA (AurA) | Aur | Other | 4b0g | A | B | 6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridine | Human | Show | |
| AURKA (AurA) | Aur | Other | 4bn1 | A | A | adenosine-5'-diphosphate | Human | Show | |
| AURKA (AurA) | Aur | Other | 4bn1 | A | B | adenosine-5'-diphosphate | Human | Show | |
| AURKA (AurA) | Aur | Other | 4byi | A | (s)-n-((1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)methyl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4byj | A | (s)-n-(1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)acetamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4c3p | A | phosphomethylphosphonic acid adenylate ester | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4c3p | D | phosphomethylphosphonic acid adenylate ester | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4c3r | A | phosphomethylphosphonic acid adenylate ester | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4ceg | A | adenosine-5'-diphosphate | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4dea | A | 4,4'-(pyrimidine-2,4-diyldiimino)dibenzoic acid | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4deb | A | 4-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4ded | A | 2-({2-[(4-carbamoylphenyl)amino]pyrimidin-4-yl}amino)benzamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4dee | A | adenosine-5'-diphosphate | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4dhf | A | 7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4dhf | B | 7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4j8m | A | 1-[4-[[4-[(5-cyclopentyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-3-[3-(trifluoromethyl)phenyl]urea | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4j8n | A | - | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4j8n | B | - | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4j8n | C | - | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4j8n | D | - | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4jai | A | n-{4-[(6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridin-1-yl)amino]phenyl}benzamide | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4jaj | A | benzo[c][1,8]naphthyridin-6(5h)-one | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4jbo | A | 1-(4-{2-[(6-{4-[2-(dimethylamino)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylurea | Human | Show | | |
| AURKA (AurA) | Aur | Other | 4jbp | A | 1-(4-{2-[(6-{4-[2-(4-hydroxypiperidin-1-yl)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylurea | Human | Show | |
