Browse kinase entries (page 169 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAP3K20 (ZAK)MLKTKL6juuAA~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamideHumanShow
MAP3K20 (ZAK)MLKTKL6juuAB~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamideHumanShow
MAP3K20 (ZAK)MLKTKL7yawAA~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamideHumanShow
MAP3K20 (ZAK)MLKTKL7yawAB~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamideHumanShow
MAP3K20 (ZAK)MLKTKL7yazAA~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamideHumanShow
MAP3K20 (ZAK)MLKTKL7yazAB~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamideHumanShow
MAP3K21 (MLK4)MLKTKL4uyaAphosphothiophosphoric acid-adenylate esterHumanShow
MAP3K5STE11STE2clqAAstaurosporineHumanShow
MAP3K5STE11STE2clqABstaurosporineHumanShow
MAP3K5STE11STE2clqBAstaurosporineHumanShow
MAP3K5STE11STE2clqBBstaurosporineHumanShow
MAP3K5STE11STE3vw6AA4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE3vw6AB4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE3vw6BA4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE3vw6BB4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE4bf2AstaurosporineHumanShow
MAP3K5STE11STE4bf2BstaurosporineHumanShow
MAP3K5STE11STE4bhnAA4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE4bhnAB4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE4bhnBA4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE4bhnBB4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHumanShow
MAP3K5STE11STE4bibAA3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHumanShow
MAP3K5STE11STE4bibAB3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHumanShow
MAP3K5STE11STE4bibBA3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHumanShow
MAP3K5STE11STE4bibBB3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHumanShow
MAP3K5STE11STE4bicAn-(2-aminoethyl)-5-{1h-pyrrolo[2,3-b]pyridin-3-yl}thiophene-2-sulfonamideHumanShow
MAP3K5STE11STE4bicB-HumanShow
MAP3K5STE11STE4bidAA5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHumanShow
MAP3K5STE11STE4bidAB5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHumanShow
MAP3K5STE11STE4bidBA5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHumanShow
MAP3K5STE11STE4bidBB5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHumanShow
MAP3K5STE11STE4bieAAn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHumanShow
MAP3K5STE11STE4bieABn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHumanShow
MAP3K5STE11STE4bieBAn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHumanShow
MAP3K5STE11STE4bieBBn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHumanShow
MAP3K5STE11STE5uorA6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHumanShow
MAP3K5STE11STE5uorB6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHumanShow
MAP3K5STE11STE5uoxA2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-oneHumanShow
MAP3K5STE11STE5uoxB2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-oneHumanShow
MAP3K5STE11STE5up3A2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHumanShow
MAP3K5STE11STE5up3B2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHumanShow
MAP3K5STE11STE5v19An-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamideHumanShow
MAP3K5STE11STE5v19Bn-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamideHumanShow
MAP3K5STE11STE5v24AA2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHumanShow
MAP3K5STE11STE5v24AB2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHumanShow
MAP3K5STE11STE5v24BA2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHumanShow
MAP3K5STE11STE5v24BB2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHumanShow
MAP3K5STE11STE5vilA2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamideHumanShow
MAP3K5STE11STE5vilB2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamideHumanShow
MAP3K5STE11STE5vilC2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamideHumanShow
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