PDB-code
Browse kinase entries (page 169 of 282)
First 165 166 167 PreviousLast173 172 171 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAP3K20 (ZAK) | MLK | TKL | 6juu | A | A | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 6juu | A | B | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 7yaw | A | A | ~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 7yaw | A | B | ~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 7yaz | A | A | ~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamide | Human | Show | ![]() |
![]() | MAP3K20 (ZAK) | MLK | TKL | 7yaz | A | B | ~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamide | Human | Show | ![]() |
![]() | MAP3K21 (MLK4) | MLK | TKL | 4uya | A | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 2clq | A | A | staurosporine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 2clq | A | B | staurosporine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 2clq | B | A | staurosporine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 2clq | B | B | staurosporine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 3vw6 | A | A | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 3vw6 | A | B | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 3vw6 | B | A | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 3vw6 | B | B | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bf2 | A | staurosporine | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 4bf2 | B | staurosporine | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 4bhn | A | A | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bhn | A | B | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bhn | B | A | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bhn | B | B | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bib | A | A | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bib | A | B | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bib | B | A | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bib | B | B | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bic | A | n-(2-aminoethyl)-5-{1h-pyrrolo[2,3-b]pyridin-3-yl}thiophene-2-sulfonamide | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 4bic | B | - | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 4bid | A | A | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bid | A | B | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bid | B | A | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bid | B | B | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bie | A | A | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bie | A | B | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bie | B | A | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 4bie | B | B | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 5uor | A | 6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5uor | B | 6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5uox | A | 2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-one | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5uox | B | 2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-one | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5up3 | A | 2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5up3 | B | 2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5v19 | A | n-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamide | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5v19 | B | n-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamide | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5v24 | A | A | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 5v24 | A | B | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 5v24 | B | A | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 5v24 | B | B | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | Show | ![]() |
![]() | MAP3K5 | STE11 | STE | 5vil | A | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5vil | B | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | Show | ![]() | |
![]() | MAP3K5 | STE11 | STE | 5vil | C | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | Show | ![]() |


