PDB-code
Browse kinase entries (page 186 of 282)
First 182 183 184 PreviousLast190 189 188 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | A | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | B | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7bdq | A | ~{n}-[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]-4-[[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]benzamide | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7be4 | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7be5 | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-methyl-pyrazole-4-carboxamide | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | A | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | B | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 7z9t | A | n-(2-cyclobutyl-1h-1,3-benzodiazol-5-yl)benzenesulfonamide | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 8acm | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 8aco | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 8aco | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 8efj | A | (4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamide | Mouse | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1a9u | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1bl6 | A | 4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazole | Human | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1bl7 | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Human | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1bmk | A | 4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazole | Human | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1di9 | A | 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline | Human | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1kv1 | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1kv2 | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | Show | ![]() | |
![]() | MAPK14 (p38a) | MAPK | CMGC | 1m7q | A | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-one | Human | Show | ![]() |


