PDB-code
Browse kinase entries (page 203 of 282)
First 199 200 201 PreviousLast207 206 205 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MERTK (MER) | Axl | TK | 7xhy | A | ~{n}-[4-(2-azanyl-3-chloranyl-pyridin-4-yl)oxy-3-fluoranyl-phenyl]-5-(4-fluorophenyl)-4-oxidanylidene-1~{h}-pyridine-3-carboxamide | Human | Show |  | |
| MET | Met | TK | 1r0p | A | k-252a | Human | Show | | |
| MET | Met | TK | 1r1w | A | - | Human | Show | | |
| MET | Met | TK | 2g15 | A | - | Human | Show | | |
| MET | Met | TK | 2rfn | A | 2-benzyl-5-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-3-methylpyrimidin-4(3h)-one | Human | Show | | |
| MET | Met | TK | 2rfn | B | 2-benzyl-5-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-3-methylpyrimidin-4(3h)-one | Human | Show | | |
| MET | Met | TK | 2rfs | A | n-(3-chlorophenyl)-n-methyl-2-oxo-3-[(3,4,5-trimethyl-1h-pyrrol-2-yl)methyl]-2h-indole-5-sulfonamide | Human | Show | | |
| MET | Met | TK | 2wd1 | A | A | 1-[(2-nitrophenyl)sulfonyl]-1h-pyrrolo[3,2-b]pyridine-6-carboxamide | Human | Show | |
| MET | Met | TK | 2wd1 | A | B | 1-[(2-nitrophenyl)sulfonyl]-1h-pyrrolo[3,2-b]pyridine-6-carboxamide | Human | Show | |
| MET | Met | TK | 2wgj | A | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | Show | | |
| MET | Met | TK | 2wkm | A | (3z)-5-[(2,6-dichlorobenzyl)sulfonyl]-3-[(3,5-dimethyl-4-{[(2s)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl}-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | Show | | |
| MET | Met | TK | 3a4p | A | (2e)-3-{6-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]quinolin-3-yl}-n-methylprop-2-enamide | Human | Show | | |
| MET | Met | TK | 3c1x | A | n-{[4-({5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}oxy)-3-fluorophenyl]carbamoyl}-2-(4-fluorophenyl)acetamide | Human | Show | | |
| MET | Met | TK | 3ccn | A | 4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]phenol | Human | Show | | |
| MET | Met | TK | 3cd8 | A | A | 7-methoxy-4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy]quinoline | Human | Show | |
| MET | Met | TK | 3cd8 | A | B | 7-methoxy-4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy]quinoline | Human | Show | |
| MET | Met | TK | 3ce3 | A | 1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | Show | | |
| MET | Met | TK | 3cth | A | n-({4-[(2-aminopyridin-4-yl)oxy]-3-fluorophenyl}carbamoyl)-2-(4-fluorophenyl)acetamide | Human | Show | | |
| MET | Met | TK | 3ctj | A | A | 2-(4-fluorophenyl)-n-{[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]carbamoyl}acetamide | Human | Show | |
| MET | Met | TK | 3ctj | A | B | 2-(4-fluorophenyl)-n-{[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]carbamoyl}acetamide | Human | Show | |
| MET | Met | TK | 3dkc | A | A | adenosine-5'-triphosphate | Human | Show | |
| MET | Met | TK | 3dkc | A | B | adenosine-5'-triphosphate | Human | Show | |
| MET | Met | TK | 3dkf | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | Show | |
| MET | Met | TK | 3dkf | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | Show | |
| MET | Met | TK | 3dkf | A | C | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | Show | |
| MET | Met | TK | 3dkg | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | Show | |
| MET | Met | TK | 3dkg | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | Show | |
| MET | Met | TK | 3dkg | A | C | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | Show | |
| MET | Met | TK | 3efj | A | 2-benzyl-5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-3-methylpyrimidin-4(3h)-one | Human | Show | | |
| MET | Met | TK | 3efj | B | 2-benzyl-5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-3-methylpyrimidin-4(3h)-one | Human | Show | | |
| MET | Met | TK | 3efk | A | 5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-2-[(4-fluorophenyl)amino]-3-methylpyrimidin-4(3h)-one | Human | Show | | |
| MET | Met | TK | 3efk | B | 5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-2-[(4-fluorophenyl)amino]-3-methylpyrimidin-4(3h)-one | Human | Show | | |
| MET | Met | TK | 3f66 | A | A | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f66 | A | B | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f66 | A | C | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f66 | A | D | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f66 | B | A | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f66 | B | B | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f66 | B | C | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f66 | B | D | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | Show | |
| MET | Met | TK | 3f82 | A | n-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorophenyl}-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | Show | | |
| MET | Met | TK | 3i5n | A | 7-methoxy-n-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]-1,5-naphthyridin-4-amine | Human | Show | | |
| MET | Met | TK | 3l8v | A | 2-({4-[(2-aminopyridin-4-yl)oxy]-3-fluorophenyl}amino)-n-(2,4-difluorophenyl)pyridine-3-carboxamide | Human | Show | | |
| MET | Met | TK | 3lq8 | A | A | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | Show | |
| MET | Met | TK | 3lq8 | A | B | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | Show | |
| MET | Met | TK | 3q6u | A | A | - | Human | Show | |
| MET | Met | TK | 3q6u | A | B | - | Human | Show | |
| MET | Met | TK | 3q6w | A | 3-{5-oxo-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-5h-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl}-n-(pyridin-2-ylmethyl)propanamide | Human | Show | | |
| MET | Met | TK | 3qti | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | Show | |
| MET | Met | TK | 3qti | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | Show | |
