Browse kinase entries (page 217 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PDPK1 (PDK1)PDK1AGC3qcsAA6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3qcsAB6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3qcxAA6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3qcxAB6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amineHumanShow
PDPK1 (PDK1)PDK1AGC3qcyAA(2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qcyAB(2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qd0AA(3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qd0AB(3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamideHumanShow
PDPK1 (PDK1)PDK1AGC3qd3AAtert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamateHumanShow
PDPK1 (PDK1)PDK1AGC3qd3ABtert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamateHumanShow
PDPK1 (PDK1)PDK1AGC3qd4AAtert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamateHumanShow
PDPK1 (PDK1)PDK1AGC3qd4ABtert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamateHumanShow
PDPK1 (PDK1)PDK1AGC3rcjA3-(1-benzyl-1h-1,2,3-triazol-4-yl)-1h-pyrrolo[2,3-b]pyridineHumanShow
PDPK1 (PDK1)PDK1AGC3rwpAA[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanoneHumanShow
PDPK1 (PDK1)PDK1AGC3rwpAB[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanoneHumanShow
PDPK1 (PDK1)PDK1AGC3rwqA[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[2-(pyridin-3-yl)ethyl]amino}pyrazin-2-yl)methanoneHumanShow
PDPK1 (PDK1)PDK1AGC3sc1A6-[2-(hydroxymethyl)phenyl]isoquinolin-1(2h)-oneHumanShow
PDPK1 (PDK1)PDK1AGC4a06AAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4a06ABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4a07AAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4a07ABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4aw0AAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4aw0ABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4aw1AAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4aw1ABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4ct1AAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4ct1ABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4ct2AAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4ct2ABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rqkAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rqkABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rqkACadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rqvAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rqvABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rqvACadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rrvAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rrvABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4rrvACadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4xx9AAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC4xx9ABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC5ackAAadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC5ackABadenosine-5'-triphosphateHumanShow
PDPK1 (PDK1)PDK1AGC5hkmA4-ethyl-6-[5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-2-amineHumanShow
PDPK1 (PDK1)PDK1AGC5hngA6-methoxy-2-(1h-pyrazol-5-yl)-1h-benzimidazoleHumanShow
PDPK1 (PDK1)PDK1AGC5ho7AA5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamideHumanShow
PDPK1 (PDK1)PDK1AGC5ho7AB5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamideHumanShow
PDPK1 (PDK1)PDK1AGC5ho8AA4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
PDPK1 (PDK1)PDK1AGC5ho8AB4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
PDPK1 (PDK1)PDK1AGC5lvlAA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHumanShow
PDPK1 (PDK1)PDK1AGC5lvlAB2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHumanShow
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