PDB-code
Browse kinase entries (page 226 of 282)
First 222 223 224 PreviousLast230 229 228 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | PIK3CG (p110g) | PIK | Atypical | 3nzs | A | 6-(1,1-dioxidothiomorpholin-4-yl)-n-(3-methoxyphenyl)-1-methyl-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show |  | |
| PIK3CG (p110g) | PIK | Atypical | 3nzu | A | 6-(2h-indazol-4-yl)-1-methyl-n-[3-(methylsulfonyl)propyl]-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3oaw | A | 2-amino-4-methyl-8-(1-methylethyl)-6-(1h-pyrazol-4-yl)pteridin-7(8h)-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3p2b | A | A | 3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenol | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 3p2b | A | B | 3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenol | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 3pre | A | 2-amino-8-(trans-4-methoxycyclohexyl)-4-methyl-6-(1h-pyrazol-3-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3prz | A | 4-amino-2-methyl-n-(1h-pyrazol-3-yl)quinazoline-8-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3ps6 | A | 4-amino-n-(6-methoxypyridin-3-yl)-2-methylquinazoline-8-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3qaq | A | [(4-{2-[(3-hydroxyphenyl)amino]-1h-benzimidazol-1-yl}-1,3,5-triazin-2-yl)amino]acetonitrile | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3qar | A | 1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-3-yl)-1h-benzimidazol-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3qjz | A | n-{6-[2-(methylsulfanyl)pyrimidin-4-yl]-1,3-benzothiazol-2-yl}acetamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3qk0 | A | n-[6-(6-chloro-5-{[(4-fluorophenyl)sulfonyl]amino}pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3r7q | A | n-(2-chlorophenyl)-n-methyl-4h-thieno[3,2-c]chromene-2-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3r7r | A | 8-(acetylamino)-n-(2-chlorophenyl)-n-methyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3s2a | A | n-{2-chloro-5-[4-(morpholin-4-yl)quinolin-6-yl]pyridin-3-yl}-4-fluorobenzenesulfonamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3sd5 | A | 5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3t8m | A | n~2~-{2-chloro-4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-n~2~,n~8~-dimethyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2,8-dicarboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3tjp | A | n~6~-(3,4-dimethoxyphenyl)-2-(morpholin-4-yl)-4,5'-bipyrimidine-2',6-diamine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3tl5 | A | (2s)-1-(4-{[2-(2-aminopyrimidin-5-yl)-7-methyl-4-(morpholin-4-yl)thieno[3,2-d]pyrimidin-6-yl]methyl}piperazin-1-yl)-2-hydroxypropan-1-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3zvv | A | 5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 3zw3 | A | n-{6-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]imidazo[1,2-a]pyridin-2-yl}acetamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4anu | A | 3-amino-n-methyl-6-[3-(1h-tetrazol-5-yl)phenyl]pyrazine-2-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4anv | A | A | 2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazine | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 4anv | A | B | 2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazine | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 4anw | A | A | 3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamide | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 4anw | A | B | 3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamide | Human | Show | |
| PIK3CG (p110g) | PIK | Atypical | 4anx | A | 5-{3-[(4-{3-[4-(1-methylethyl)phenyl]pyrazin-2-yl}piperazin-1-yl)sulfonyl]phenyl}pyrimidin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4aof | A | n-[6-(5-methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]ethanamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4dk5 | A | 4-(2-[(6-methoxypyridin-3-yl)amino]-5-{[4-(methylsulfonyl)piperazin-1-yl]methyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4ezj | A | 2-(1-{[2-(5-fluoro-1h-indol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4ezk | A | 2-(1-{[2-(2h-indazol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4ezl | A | 2-(1-{[2-(2-aminopyrimidin-5-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4f1s | A | n-(5-{[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(tetrahydro-2h-pyran-4-yl)pyridin-2-yl]amino}-2-chloropyridin-3-yl)methanesulfonamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4fa6 | A | 2-amino-8-cyclopentyl-4-methyl-6-(1h-pyrazol-4-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4fad | A | 2-amino-6-(5-fluoro-6-methoxypyridin-3-yl)-4-methyl-8-(pyrrolidin-1-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4fhj | A | 3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-5-yl)imidazo[1,2-a]pyridin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4fhk | A | 3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]-n-(1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4fjy | A | 4-[3,3-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1h-indol-1-yl]-7-fluoro-3-methyl-2-(pyridin-3-yl)quinoline | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4fjz | A | 1'-[7-fluoro-3-methyl-2-(pyridin-2-yl)quinolin-4-yl]-6'-(morpholin-4-yl)-1',2,2',3,5,6-hexahydrospiro[pyran-4,3'-pyrrolo[3,2-b]pyridine] | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4flh | A | 4-(2-[(5-fluoro-6-methoxypyridin-3-yl)amino]-5-{(1r)-1-[4-(methylsulfonyl)piperazin-1-yl]ethyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amine | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4ful | A | 4-({4-[3-(piperidin-1-ylcarbonyl)phenyl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4g11 | A | 2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]-n-phenylacetamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4gb9 | A | 2-[1-({2-[2-(dimethylamino)-1h-benzimidazol-1-yl]-9-methyl-6-(morpholin-4-yl)-9h-purin-8-yl}methyl)piperidin-4-yl]propan-2-ol | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4hle | A | 2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepine-8-carboxamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4hvb | A | 1-{1-[(2s)-2-hydroxypropanoyl]piperidin-4-yl}-3-methyl-8-(6-methylpyridin-3-yl)-1,3-dihydro-2h-imidazo[4,5-c][1,5]naphthyridin-2-one | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4j6i | A | 2-methyl-1-(4-{2-[1-(2,2,2-trifluoroethyl)-1h-1,2,4-triazol-5-yl]-4,5-dihydro[1]benzoxepino[5,4-d][1,3]thiazol-8-yl}-1h-pyrazol-1-yl)propan-2-ol | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4kz0 | A | methyl 2-(acetylamino)-1,3-benzothiazole-6-carboxylate | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4kzc | A | n-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamide | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4ps3 | A | 1-[6-(5-methoxypyridin-3-yl)-1,3-benzothiazol-2-yl]-3-[2-(1-propyl-1h-imidazol-4-yl)ethyl]urea | Human | Show | | |
| PIK3CG (p110g) | PIK | Atypical | 4ps7 | A | n-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | Show | |
