PDB-code
Browse kinase entries (page 265 of 282)
First 261 262 263 PreviousLast269 268 267 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | TEK (TIE2) | Tie | TK | 1fvr | B | - | Human | Show |  | |
| TEK (TIE2) | Tie | TK | 2oo8 | X | n-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)phenyl}-4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]benzamide | Human | Show | | |
| TEK (TIE2) | Tie | TK | 2osc | A | n-{4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]phenyl}-3-(trifluoromethyl)benzamide | Human | Show | | |
| TEK (TIE2) | Tie | TK | 2p4i | A | 4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamide | Human | Show | | |
| TEK (TIE2) | Tie | TK | 2p4i | B | 4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamide | Human | Show | | |
| TEK (TIE2) | Tie | TK | 2wqb | A | 2-[3-(cyclohexylmethyl)-5-phenyl-imidazol-4-yl]-[1,3]thiazolo[4,5-e]pyrimidin-7-amine | Human | Show | | |
| TEK (TIE2) | Tie | TK | 3l8p | A | 2-methyl-11-(1-methylethyl)-8-[(2s)-tetrahydro-2h-pyran-2-yl]-2,11,12,13-tetrahydro-4h-indazolo[5,4-a]pyrrolo[3,4-c]carbazol-4-one | Human | Show | | |
| TEK (TIE2) | Tie | TK | 4x3j | A | 1-[4-(4-amino-5-oxopyrido[2,3-d]pyrimidin-8(5h)-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | Human | Show | | |
| TEK (TIE2) | Tie | TK | 6mwe | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
| TEK (TIE2) | Tie | TK | 6mwe | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
| TEK (TIE2) | Tie | TK | 6mwe | B | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
| TEK (TIE2) | Tie | TK | 6mwe | B | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | B | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | D | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | F | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | H | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | A | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | B | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | C | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | D | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | E | - | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1py5 | A | 4-(3-pyridin-2-yl-1h-pyrazol-4-yl)quinoline | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1rw8 | A | 3-(4-fluorophenyl)-2-(6-methylpyridin-2-yl)-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazole | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1vjy | A | 2-[5-(6-methylpyridin-2-yl)-2,3-dihydro-1h-pyrazol-4-yl]-1,5-naphthyridine | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | A | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | B | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wou | A | 4-({4-[(2,6-dimethylpyridin-3-yl)oxy]pyridin-2-yl}amino)benzenesulfonamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | A | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | B | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | C | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | D | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | E | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | A | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | B | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | C | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | D | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | E | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3gxl | A | n-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amine | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3hmm | A | 2-(6-methylpyridin-2-yl)-n-pyridin-4-ylquinazolin-4-amine | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | A | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | B | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | C | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | D | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | E | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | A | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | B | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | A | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | B | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | A | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | Show | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | B | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | Show | |
