PDB-code
Browse kinase entries (page 268 of 282)
First 264 265 266 PreviousLast272 271 270 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | TNK2 (ACK) | Ack | TK | 5zxb | A | A | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 5zxb | A | B | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 5zxb | B | A | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 5zxb | B | B | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 6vqm | A | 2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-one | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 6vqm | B | 2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-one | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 7kp6 | A | A | 5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 7kp6 | A | B | 5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 8fe9 | A | n-[(1s)-1-benzyl-2-[(6-chloro-2-oxo-1h-quinolin-4-yl)methylamino]-2-oxo-ethyl]-4-hydroxy-2-oxo-1h-quinoline-6-carbo | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 8hmt | A | A | 6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-one | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 8hmt | A | B | 6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-one | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | A | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | A | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | B | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | B | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | C | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | C | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | D | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | D | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | A | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | A | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | B | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | B | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | C | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | C | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | D | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | D | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | A | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | A | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | A | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | B | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | B | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | B | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | C | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | C | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | C | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | D | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | D | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | D | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 7mgj | A | n-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamide | Human | Show | ![]() | |
![]() | TNNI3K (HH498) | MLK | TKL | 7mgk | A | A | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 7mgk | A | B | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | Show | ![]() |
![]() | TP53RK (PRPK) | Bud32 | Other | 6wqx | C | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | TP53RK (PRPK) | Bud32 | Other | 6wqx | D | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | TP53RK (PRPK) | Bud32 | Other | 7sza | A | A | 4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | Show | ![]() |
![]() | TP53RK (PRPK) | Bud32 | Other | 7sza | A | B | 4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | Show | ![]() |
![]() | TP53RK (PRPK) | Bud32 | Other | 7szb | A | 5-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | Show | ![]() | |
![]() | TP53RK (PRPK) | Bud32 | Other | 7szc | A | 4-hydroxy-2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | Show | ![]() | |
![]() | TP53RK (PRPK) | Bud32 | Other | 7szd | A | 2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1,3-dioxo-2,3-dihydro-1h-isoindole-5-carboxylic acid | Human | Show | ![]() | |
![]() | TRIB1 (Trb1) | Trbl | CAMK | 5cek | A | - | Human | Show | ![]() |


