Browse kinase entries (page 268 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
TNK2 (ACK)AckTK5zxbAAn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHumanShow
TNK2 (ACK)AckTK5zxbABn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHumanShow
TNK2 (ACK)AckTK5zxbBAn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHumanShow
TNK2 (ACK)AckTK5zxbBBn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHumanShow
TNK2 (ACK)AckTK6vqmA2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-oneHumanShow
TNK2 (ACK)AckTK6vqmB2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-oneHumanShow
TNK2 (ACK)AckTK7kp6AA5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamineHumanShow
TNK2 (ACK)AckTK7kp6AB5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamineHumanShow
TNK2 (ACK)AckTK8fe9An-[(1s)-1-benzyl-2-[(6-chloro-2-oxo-1h-quinolin-4-yl)methylamino]-2-oxo-ethyl]-4-hydroxy-2-oxo-1h-quinoline-6-carboHumanShow
TNK2 (ACK)AckTK8hmtAA6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-oneHumanShow
TNK2 (ACK)AckTK8hmtAB6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-oneHumanShow
TNNI3K (HH498)MLKTKL4yffAA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yffAB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yffBA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yffBB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yffCA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yffCB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yffDA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yffDB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiAAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiABn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiBAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiBBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiCAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiCBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiDAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL4yfiDBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jAAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jABn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jACn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jBAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jBBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jBCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jCAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jCBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jCCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jDAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jDBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL6b5jDCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHumanShow
TNNI3K (HH498)MLKTKL7mgjAn-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamideHumanShow
TNNI3K (HH498)MLKTKL7mgkAAn-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]ureaHumanShow
TNNI3K (HH498)MLKTKL7mgkABn-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]ureaHumanShow
TP53RK (PRPK)Bud32Other6wqxCphosphoaminophosphonic acid-adenylate esterHumanShow
TP53RK (PRPK)Bud32Other6wqxDphosphoaminophosphonic acid-adenylate esterHumanShow
TP53RK (PRPK)Bud32Other7szaAA4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHumanShow
TP53RK (PRPK)Bud32Other7szaAB4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHumanShow
TP53RK (PRPK)Bud32Other7szbA5-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHumanShow
TP53RK (PRPK)Bud32Other7szcA4-hydroxy-2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHumanShow
TP53RK (PRPK)Bud32Other7szdA2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1,3-dioxo-2,3-dihydro-1h-isoindole-5-carboxylic acidHumanShow
TRIB1 (Trb1)TrblCAMK5cekA-HumanShow
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