PDB-code
Browse kinase entries (page 274 of 282)
First 270 271 272 PreviousLast278 277 276 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | ULK1 | ULK | Other | 4wno | A | A | n~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wno | A | B | n~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | A | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | A | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | B | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | B | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | C | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | C | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | D | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 4wnp | D | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 5ci7 | A | A | n-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 5ci7 | A | B | n-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 6mnh | A | A | n-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 6mnh | A | B | n-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 6qas | A | A | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 6qas | A | B | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 6qas | B | A | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 6qas | B | B | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 8sv9 | A | A | (4p)-4-[(2p)-2-(1,2,5,6-tetrahydropyridin-3-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n-(2,2,2-trifluoroethyl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | ULK1 | ULK | Other | 8sv9 | A | B | (4p)-4-[(2p)-2-(1,2,5,6-tetrahydropyridin-3-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n-(2,2,2-trifluoroethyl)thiophene-2-carboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qat | A | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | Show | ![]() | |
![]() | ULK2 | ULK | Other | 6qat | B | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | Show | ![]() | |
![]() | ULK2 | ULK | Other | 6qat | C | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | Show | ![]() | |
![]() | ULK2 | ULK | Other | 6qat | D | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | Show | ![]() | |
![]() | ULK2 | ULK | Other | 6qau | A | A | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qau | A | B | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qau | B | A | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qau | B | B | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qau | C | A | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qau | C | B | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | A | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | A | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | B | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | B | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | C | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | C | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | D | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6qav | D | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | A | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | A | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | B | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | B | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | C | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | C | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | D | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK2 | ULK | Other | 6yid | D | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | Show | ![]() |
![]() | ULK3 | ULK | Other | 6fdy | U | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | ![]() | |
![]() | ULK3 | ULK | Other | 6fdz | U | momelotinib | Human | Show | ![]() | |
![]() | ULK4 | ULK | Other | 6tsz | U | phosphothiophosphoric acid-adenylate ester | Human | Show | ![]() | |
![]() | ULK4 | ULK | Other | 6u5l | A | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | Show | ![]() |


