PDB-code
Browse kinase entries (page 278 of 282)
First 274 275 276 PreviousLast281 280 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | VRK1 | VRK | CK1 | 6cmm | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show |  |
| VRK1 | VRK | CK1 | 6cnx | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cnx | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cnx | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cnx | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cnx | C | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cnx | C | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cnx | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cnx | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | C | A | - | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | C | B | - | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6cqh | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | A | A | - | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | A | B | - | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | B | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | B | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | C | A | - | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | C | B | - | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | D | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6csw | D | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | A | A | - | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | A | B | - | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | C | A | - | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | C | B | - | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6dd4 | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | Show | |
| VRK1 | VRK | CK1 | 6npn | A | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| VRK1 | VRK | CK1 | 6npn | B | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| VRK1 | VRK | CK1 | 6npn | C | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| VRK1 | VRK | CK1 | 6npn | D | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| VRK1 | VRK | CK1 | 6vxu | B | (7r)-8-(cyclopropylmethyl)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| VRK1 | VRK | CK1 | 6vzh | A | - | Human | Show | | |
| VRK1 | VRK | CK1 | 6vzh | B | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | Show | | |
| VRK1 | VRK | CK1 | 6vzh | C | - | Human | Show | | |
| VRK1 | VRK | CK1 | 6vzh | D | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | Show | | |
| VRK1 | VRK | CK1 | 8v42 | A | A | - | Human | Show | |
| VRK1 | VRK | CK1 | 8v42 | A | B | - | Human | Show | |
| VRK2 | VRK | CK1 | 2v62 | A | A | - | Human | Show | |
| VRK2 | VRK | CK1 | 2v62 | A | B | - | Human | Show | |
| VRK2 | VRK | CK1 | 2v62 | B | A | - | Human | Show | |
| VRK2 | VRK | CK1 | 2v62 | B | B | - | Human | Show | |
| VRK2 | VRK | CK1 | 5uu1 | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| VRK2 | VRK | CK1 | 6ncg | A | 4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamide | Human | Show | |
