Browse kinase entries (page 40 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC1vyzAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzamideHumanShow
CDK2CDKCMGC1w0xCAolomoucineHumanShow
CDK2CDKCMGC1w0xCBolomoucineHumanShow
CDK2CDKCMGC1w8cAA6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHumanShow
CDK2CDKCMGC1w8cAB6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHumanShow
CDK2CDKCMGC1w98A-HumanShow
CDK2CDKCMGC1wccAA2-amino-6-chloropyrazineHumanShow
CDK2CDKCMGC1wccAB2-amino-6-chloropyrazineHumanShow
CDK2CDKCMGC1y8yA(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amineHumanShow
CDK2CDKCMGC1y91A4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamideHumanShow
CDK2CDKCMGC1ykrA4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC2a0cXA2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHumanShow
CDK2CDKCMGC2a0cXB2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHumanShow
CDK2CDKCMGC2a4lAr-roscovitineHumanShow
CDK2CDKCMGC2b52A1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)ureaHumanShow
CDK2CDKCMGC2b53A6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amineHumanShow
CDK2CDKCMGC2b54A6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-oneHumanShow
CDK2CDKCMGC2b55A2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamideHumanShow
CDK2CDKCMGC2bheA(2z)-5'-bromo-2,3'-biindole-2',3(1h,1'h)-dione ammoniateHumanShow
CDK2CDKCMGC2bhhA(2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-oneHumanShow
CDK2CDKCMGC2bkzA1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHumanShow
CDK2CDKCMGC2bkzC1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHumanShow
CDK2CDKCMGC2bpmA(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHumanShow
CDK2CDKCMGC2bpmC(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHumanShow
CDK2CDKCMGC2btrAn-(5-isopropyl-thiazol-2-yl)-2-pyridin-3-yl-acetamideHumanShow
CDK2CDKCMGC2btsA4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHumanShow
CDK2CDKCMGC2c4gA(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHumanShow
CDK2CDKCMGC2c4gC(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHumanShow
CDK2CDKCMGC2c5nAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHumanShow
CDK2CDKCMGC2c5nABn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHumanShow
CDK2CDKCMGC2c5nCAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHumanShow
CDK2CDKCMGC2c5nCBn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHumanShow
CDK2CDKCMGC2c5oAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5oAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5oCA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5oCB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5vAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5vAB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5vCA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5vCB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHumanShow
CDK2CDKCMGC2c5xAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHumanShow
CDK2CDKCMGC2c5xABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHumanShow
CDK2CDKCMGC2c5xCAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHumanShow
CDK2CDKCMGC2c5xCBhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHumanShow
CDK2CDKCMGC2c5yAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHumanShow
CDK2CDKCMGC2c5yABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHumanShow
CDK2CDKCMGC2c68A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2c69A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2c6iA4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC2c6kA4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHumanShow
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