Browse kinase entries (page 44 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC3bhtAB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC3bhtCA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC3bhtCB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC3bhuAA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC3bhuAB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC3bhuCA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC3bhuCB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC3bhvAA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHumanShow
CDK2CDKCMGC3bhvAB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHumanShow
CDK2CDKCMGC3bhvCA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHumanShow
CDK2CDKCMGC3bhvCB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHumanShow
CDK2CDKCMGC3ddpAA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHumanShow
CDK2CDKCMGC3ddpAB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHumanShow
CDK2CDKCMGC3ddpCA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHumanShow
CDK2CDKCMGC3ddpCB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHumanShow
CDK2CDKCMGC3ddqAAr-roscovitineHumanShow
CDK2CDKCMGC3ddqABr-roscovitineHumanShow
CDK2CDKCMGC3ddqCAr-roscovitineHumanShow
CDK2CDKCMGC3ddqCBr-roscovitineHumanShow
CDK2CDKCMGC3dogAA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHumanShow
CDK2CDKCMGC3dogAB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHumanShow
CDK2CDKCMGC3dogCA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHumanShow
CDK2CDKCMGC3dogCB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHumanShow
CDK2CDKCMGC3eidAA(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHumanShow
CDK2CDKCMGC3eidAB(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHumanShow
CDK2CDKCMGC3eidCA-HumanShow
CDK2CDKCMGC3eidCB-HumanShow
CDK2CDKCMGC3ej1An-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHumanShow
CDK2CDKCMGC3ej1Cn-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHumanShow
CDK2CDKCMGC3eocA5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHumanShow
CDK2CDKCMGC3eocC5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHumanShow
CDK2CDKCMGC3ezrA3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHumanShow
CDK2CDKCMGC3ezvA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHumanShow
CDK2CDKCMGC3f5xA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHumanShow
CDK2CDKCMGC3f5xC4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHumanShow
CDK2CDKCMGC3fz1A(3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-oneHumanShow
CDK2CDKCMGC3ig7An-{1-[cis-3-(acetylamino)cyclobutyl]-1h-imidazol-4-yl}-2-(4-methoxyphenyl)acetamideHumanShow
CDK2CDKCMGC3iggAn-[1-(cis-3-hydroxycyclobutyl)-1h-imidazol-4-yl]-2-(4-methoxyphenyl)acetamideHumanShow
CDK2CDKCMGC3le6A5-(2-chlorophenyl)-3-methyl-7-nitropyrazolo[3,4-b][1,4]benzodiazepineHumanShow
CDK2CDKCMGC3lfnAn-[6-(4-hydroxyphenyl)-5-phenyl-1h-indazol-3-yl]butanamideHumanShow
CDK2CDKCMGC3lfqAn-(6,7-difluoro-5-phenyl-1h-indazol-3-yl)butanamideHumanShow
CDK2CDKCMGC3lfsAn-(6-chloro-5-phenyl-1h-indazol-3-yl)butanamideHumanShow
CDK2CDKCMGC3my5AA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHumanShow
CDK2CDKCMGC3my5AB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHumanShow
CDK2CDKCMGC3my5AC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHumanShow
CDK2CDKCMGC3my5CA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHumanShow
CDK2CDKCMGC3my5CB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHumanShow
CDK2CDKCMGC3my5CC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHumanShow
CDK2CDKCMGC3ns9A(2s,3s)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triolHumanShow
CDK2CDKCMGC3pj8AA(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHumanShow
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