PDB-code
Browse kinase entries (page 47 of 282)
First 43 44 45 PreviousLast51 50 49 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CDK2 | CDK | CMGC | 3r8p | A | A | (5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r8p | A | B | (5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r8u | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r8u | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r8v | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r8v | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r8z | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r8z | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r9d | A | A | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r9d | A | B | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r9h | A | A | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r9h | A | B | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r9n | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r9n | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3r9o | A | 4-amino-n-(3,5-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 3rah | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rah | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rai | A | A | 4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rai | A | B | 4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rak | A | A | 4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rak | A | B | 4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3ral | A | A | 4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3ral | A | B | 4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rjc | A | A | {4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rjc | A | B | {4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rk5 | A | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzoic acid | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 3rk7 | A | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 3rk9 | A | A | [4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rk9 | A | B | [4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rkb | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rkb | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rm6 | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rm6 | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rm7 | A | A | 2-[(4-hydroxybenzyl)amino]-5-nitrobenzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rm7 | A | B | 2-[(4-hydroxybenzyl)amino]-5-nitrobenzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rmf | A | A | 4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rmf | A | B | 4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rni | A | A | 3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rni | A | B | 3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3roy | A | A | 4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3roy | A | B | 4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpo | A | A | 4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpo | A | B | 4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpr | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpr | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpv | A | A | 4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpv | A | B | 4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpy | A | A | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rpy | A | B | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 3rzb | A | A | 4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamide | Human | Show | ![]() |


