Browse kinase entries (page 51 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC4fkiABn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHumanShow
CDK2CDKCMGC4fkjAAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHumanShow
CDK2CDKCMGC4fkjABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHumanShow
CDK2CDKCMGC4fklAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC4fklAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHumanShow
CDK2CDKCMGC4fkoAA2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHumanShow
CDK2CDKCMGC4fkoAB2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHumanShow
CDK2CDKCMGC4fkpAA3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHumanShow
CDK2CDKCMGC4fkpAB3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHumanShow
CDK2CDKCMGC4fkpAC3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHumanShow
CDK2CDKCMGC4fkqAA4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHumanShow
CDK2CDKCMGC4fkqAB4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHumanShow
CDK2CDKCMGC4fkrAA(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHumanShow
CDK2CDKCMGC4fkrAB(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHumanShow
CDK2CDKCMGC4fksAAn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHumanShow
CDK2CDKCMGC4fksABn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHumanShow
CDK2CDKCMGC4fksACn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHumanShow
CDK2CDKCMGC4fktAAn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC4fktABn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC4fkuAA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHumanShow
CDK2CDKCMGC4fkuAB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHumanShow
CDK2CDKCMGC4fkvAA(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHumanShow
CDK2CDKCMGC4fkvAB(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHumanShow
CDK2CDKCMGC4fkwAA2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHumanShow
CDK2CDKCMGC4fkwAB2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHumanShow
CDK2CDKCMGC4fx3AA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHumanShow
CDK2CDKCMGC4fx3AB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHumanShow
CDK2CDKCMGC4fx3CA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHumanShow
CDK2CDKCMGC4fx3CB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHumanShow
CDK2CDKCMGC4gcjAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC4gcjAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC4i3zAadenosine-5'-diphosphateHumanShow
CDK2CDKCMGC4i3zCadenosine-5'-diphosphateHumanShow
CDK2CDKCMGC4ii5AAadenosine-5'-diphosphateHumanShow
CDK2CDKCMGC4ii5ABadenosine-5'-diphosphateHumanShow
CDK2CDKCMGC4ii5CAadenosine-5'-diphosphateHumanShow
CDK2CDKCMGC4ii5CBadenosine-5'-diphosphateHumanShow
CDK2CDKCMGC4kd1AA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHumanShow
CDK2CDKCMGC4kd1AB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHumanShow
CDK2CDKCMGC4lynA(2s)-n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)-2-phenylpropanamideHumanShow
CDK2CDKCMGC4nj3AA6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHumanShow
CDK2CDKCMGC4nj3AB6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHumanShow
CDK2CDKCMGC4rj3AA1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHumanShow
CDK2CDKCMGC4rj3AB1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHumanShow
CDK2CDKCMGC5a14AA1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHumanShow
CDK2CDKCMGC5a14AB1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHumanShow
CDK2CDKCMGC5andA2-imidazol-1-yl-1h-benzimidazoleHumanShow
CDK2CDKCMGC5aneA6-methoxy-9h-purineHumanShow
CDK2CDKCMGC5angA7-hydroxy-4-(morpholinomethyl)chromen-2-oneHumanShow
CDK2CDKCMGC5aniA6-chloro-9h-purineHumanShow
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