Browse kinase entries (page 55 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC7s7aAA2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7s7aAB2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7s84AA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7s84AB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7s85A2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethoxy)benzoic acidHumanShow
CDK2CDKCMGC7s9xAA2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7s9xAB2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7sa0AA2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7sa0AB2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHumanShow
CDK2CDKCMGC7ug1AA8-(4-chloroanilino)naphthalene-1-sulfonic acidHumanShow
CDK2CDKCMGC7ug1AB8-(4-chloroanilino)naphthalene-1-sulfonic acidHumanShow
CDK2CDKCMGC7uxiAA-HumanShow
CDK2CDKCMGC7uxiAB-HumanShow
CDK2CDKCMGC7uxkA-HumanShow
CDK2CDKCMGC7vduAA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHumanShow
CDK2CDKCMGC7vduAB[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHumanShow
CDK2CDKCMGC7zpcAA~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHumanShow
CDK2CDKCMGC7zpcAB~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHumanShow
CDK2CDKCMGC8b54AA~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHumanShow
CDK2CDKCMGC8b54AB~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHumanShow
CDK2CDKCMGC8byaA-HumanShow
CDK2CDKCMGC8bzoA-HumanShow
CDK2CDKCMGC8curAA6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHumanShow
CDK2CDKCMGC8curAB6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHumanShow
CDK2CDKCMGC8erdAA(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHumanShow
CDK2CDKCMGC8erdAB(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHumanShow
CDK2CDKCMGC8ernAAn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHumanShow
CDK2CDKCMGC8ernABn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHumanShow
CDK2CDKCMGC8fowAA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHumanShow
CDK2CDKCMGC8fowAB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHumanShow
CDK2CDKCMGC8fp0AAr-roscovitineHumanShow
CDK2CDKCMGC8fp0ABr-roscovitineHumanShow
CDK2CDKCMGC8fp5AAadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC8fp5ABadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC8h6pA(7s,10r)-11-oxa-2,4,5,13,17,23-hexaazatetracyclo[17.3.1.1~3,6~.1~7,10~]pentacosa-1(23),3(25),5,19,21-pentaene-12,18-dioneHumanShow
CDK2CDKCMGC8h6tA(1r,3s)-3-{3-[(pyridin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl propan-2-ylcarbamateHumanShow
CDK2CDKCMGC8oy2A(1s,2s,11as)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dioneHumanShow
CDK2CDKCMGC8ru8AA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK2CDKCMGC8ru8AB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK2CDKCMGC8uv0AA1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-olHumanShow
CDK2CDKCMGC8uv0AB1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-olHumanShow
CDK4CDKCMGC2w96BA-HumanShow
CDK4CDKCMGC2w96BB-HumanShow
CDK4CDKCMGC2w99B-HumanShow
CDK4CDKCMGC2w9fB-HumanShow
CDK4CDKCMGC2w9zBA-HumanShow
CDK4CDKCMGC2w9zBB-HumanShow
CDK4CDKCMGC3g33A-HumanShow
CDK4CDKCMGC3g33C-HumanShow
CDK4CDKCMGC5fwkK-HumanShow
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