PDB-code
Browse kinase entries (page 55 of 282)
First 51 52 53 PreviousLast59 58 57 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CDK2 | CDK | CMGC | 7s7a | A | A | 2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7s7a | A | B | 2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7s84 | A | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7s84 | A | B | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7s85 | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethoxy)benzoic acid | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7s9x | A | A | 2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7s9x | A | B | 2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7sa0 | A | A | 2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7sa0 | A | B | 2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ug1 | A | A | 8-(4-chloroanilino)naphthalene-1-sulfonic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7ug1 | A | B | 8-(4-chloroanilino)naphthalene-1-sulfonic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7uxi | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7uxi | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7uxk | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 7vdu | A | A | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7vdu | A | B | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7zpc | A | A | ~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 7zpc | A | B | ~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8b54 | A | A | ~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8b54 | A | B | ~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8bya | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 8bzo | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 8cur | A | A | 6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8cur | A | B | 6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8erd | A | A | (2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8erd | A | B | (2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8ern | A | A | n,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8ern | A | B | n,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamide | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8fow | A | A | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8fow | A | B | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8fp0 | A | A | r-roscovitine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8fp0 | A | B | r-roscovitine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8fp5 | A | A | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8fp5 | A | B | adenosine-5'-triphosphate | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8h6p | A | (7s,10r)-11-oxa-2,4,5,13,17,23-hexaazatetracyclo[17.3.1.1~3,6~.1~7,10~]pentacosa-1(23),3(25),5,19,21-pentaene-12,18-dione | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 8h6t | A | (1r,3s)-3-{3-[(pyridin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl propan-2-ylcarbamate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 8oy2 | A | (1s,2s,11as)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dione | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 8ru8 | A | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8ru8 | A | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8uv0 | A | A | 1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 8uv0 | A | B | 1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-ol | Human | Show | ![]() |
![]() | CDK4 | CDK | CMGC | 2w96 | B | A | - | Human | Show | ![]() |
![]() | CDK4 | CDK | CMGC | 2w96 | B | B | - | Human | Show | ![]() |
![]() | CDK4 | CDK | CMGC | 2w99 | B | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 2w9f | B | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 2w9z | B | A | - | Human | Show | ![]() |
![]() | CDK4 | CDK | CMGC | 2w9z | B | B | - | Human | Show | ![]() |
![]() | CDK4 | CDK | CMGC | 3g33 | A | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 3g33 | C | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 5fwk | K | - | Human | Show | ![]() |


