PDB-code
Browse kinase entries (page 56 of 282)
First 52 53 54 PreviousLast60 59 58 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CDK4 | CDK | CMGC | 5fwl | K | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 5fwm | K | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 5fwp | K | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 6p8e | B | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 6p8f | B | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 6p8g | B | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 6p8h | B | - | Human | Show | ![]() | |
![]() | CDK4 | CDK | CMGC | 7sj3 | A | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1h4l | A | - | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1h4l | B | - | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1ung | A | 6-phenyl[5h]pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1ung | B | 6-phenyl[5h]pyrrolo[2,3-b]pyrazine | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1unh | A | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1unh | B | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1unl | A | r-roscovitine | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 1unl | B | - | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 3o0g | A | - | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 3o0g | B | {4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanone | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 4au8 | A | A | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | CDK5 | CDK | CMGC | 4au8 | A | B | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | CDK5 | CDK | CMGC | 4au8 | B | A | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | CDK5 | CDK | CMGC | 4au8 | B | B | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | Show | ![]() |
![]() | CDK5 | CDK | CMGC | 7vdp | A | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 7vdq | A | 2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acid | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 7vdr | A | (1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanol | Human | Show | ![]() | |
![]() | CDK5 | CDK | CMGC | 7vds | A | A | 5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrile | Human | Show | ![]() |
![]() | CDK5 | CDK | CMGC | 7vds | A | B | 5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrile | Human | Show | ![]() |
![]() | CDK6 | CDK | CMGC | 1bi7 | A | - | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 1bi8 | A | - | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 1bi8 | C | - | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 1blx | A | - | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 1g3n | A | - | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 1g3n | E | - | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 1jow | B | - | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 1xo2 | B | 3,7,3',4'-tetrahydroxyflavone | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 2euf | B | 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 2f2c | B | (2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 3nup | A | 4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 3nux | A | 4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 4aua | A | 1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanone | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 4ez5 | A | {5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanone | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 4tth | B | 9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 5l2i | A | 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 5l2s | A | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 5l2t | A | 7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 6oql | A | 5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 6oqo | A | n-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK6 | CDK | CMGC | 8i0m | A | 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | Show | ![]() | |
![]() | CDK7 | CDK | CMGC | 1ua2 | A | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK7 | CDK | CMGC | 1ua2 | B | adenosine-5'-triphosphate | Human | Show | ![]() |


