Browse kinase entries (page 56 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK4CDKCMGC5fwlK-HumanShow
CDK4CDKCMGC5fwmK-HumanShow
CDK4CDKCMGC5fwpK-HumanShow
CDK4CDKCMGC6p8eB-HumanShow
CDK4CDKCMGC6p8fB-HumanShow
CDK4CDKCMGC6p8gB-HumanShow
CDK4CDKCMGC6p8hB-HumanShow
CDK4CDKCMGC7sj3An-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHumanShow
CDK5CDKCMGC1h4lA-HumanShow
CDK5CDKCMGC1h4lB-HumanShow
CDK5CDKCMGC1ungA6-phenyl[5h]pyrrolo[2,3-b]pyrazineHumanShow
CDK5CDKCMGC1ungB6-phenyl[5h]pyrrolo[2,3-b]pyrazineHumanShow
CDK5CDKCMGC1unhA(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHumanShow
CDK5CDKCMGC1unhB(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHumanShow
CDK5CDKCMGC1unlAr-roscovitineHumanShow
CDK5CDKCMGC1unlB-HumanShow
CDK5CDKCMGC3o0gA-HumanShow
CDK5CDKCMGC3o0gB{4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanoneHumanShow
CDK5CDKCMGC4au8AA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow
CDK5CDKCMGC4au8AB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow
CDK5CDKCMGC4au8BA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow
CDK5CDKCMGC4au8BB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow
CDK5CDKCMGC7vdpA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHumanShow
CDK5CDKCMGC7vdqA2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acidHumanShow
CDK5CDKCMGC7vdrA(1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanolHumanShow
CDK5CDKCMGC7vdsAA5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHumanShow
CDK5CDKCMGC7vdsAB5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHumanShow
CDK6CDKCMGC1bi7A-HumanShow
CDK6CDKCMGC1bi8A-HumanShow
CDK6CDKCMGC1bi8C-HumanShow
CDK6CDKCMGC1blxA-HumanShow
CDK6CDKCMGC1g3nA-HumanShow
CDK6CDKCMGC1g3nE-HumanShow
CDK6CDKCMGC1jowB-HumanShow
CDK6CDKCMGC1xo2B3,7,3',4'-tetrahydroxyflavoneHumanShow
CDK6CDKCMGC2eufB6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHumanShow
CDK6CDKCMGC2f2cB(2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHumanShow
CDK6CDKCMGC3nupA4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amineHumanShow
CDK6CDKCMGC3nuxA4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineHumanShow
CDK6CDKCMGC4auaA1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanoneHumanShow
CDK6CDKCMGC4ez5A{5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanoneHumanShow
CDK6CDKCMGC4tthB9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amineHumanShow
CDK6CDKCMGC5l2iA6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHumanShow
CDK6CDKCMGC5l2sAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHumanShow
CDK6CDKCMGC5l2tA7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHumanShow
CDK6CDKCMGC6oqlA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHumanShow
CDK6CDKCMGC6oqoAn-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHumanShow
CDK6CDKCMGC8i0mA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHumanShow
CDK7CDKCMGC1ua2Aadenosine-5'-triphosphateHumanShow
CDK7CDKCMGC1ua2Badenosine-5'-triphosphateHumanShow
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