Browse kinase entries (page 59 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK9CDKCMGC8i0lA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHumanShow
CDK9CDKCMGC8k5rA(1s,3s)-n3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamineHumanShow
CDKL1CDKLCMGC4aguAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
CDKL1CDKLCMGC4aguBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
CDKL1CDKLCMGC4aguCn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
CDKL2CDKLCMGC4aaaAA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHumanShow
CDKL2CDKLCMGC4aaaAB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHumanShow
CDKL2CDKLCMGC4bbmA4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diolHumanShow
CDKL2CDKLCMGC4bbmB4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diolHumanShow
CDKL3CDKLCMGC3zduA[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHumanShow
CDKL5CDKLCMGC4bgqAA[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHumanShow
CDKL5CDKLCMGC4bgqAB[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHumanShow
CDKL5CDKLCMGC8cieA4-[[3,5-bis(fluoranyl)phenyl]carbonylamino]-~{n}-piperidin-4-yl-1~{h}-pyrazole-3-carboxamideHumanShow
CHEK1 (CHK1)CAMKLCAMK1ia8A-HumanShow
CHEK1 (CHK1)CAMKLCAMK1nvqA7-hydroxystaurosporineHumanShow
CHEK1 (CHK1)CAMKLCAMK1nvrAstaurosporineHumanShow
CHEK1 (CHK1)CAMKLCAMK1nvsArel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dioneHumanShow
CHEK1 (CHK1)CAMKLCAMK1zltA(4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK1zysAn-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamideHumanShow
CHEK1 (CHK1)CAMKLCAMK2aypA(3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2br1AA2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHumanShow
CHEK1 (CHK1)CAMKLCAMK2br1AB2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHumanShow
CHEK1 (CHK1)CAMKLCAMK2brbA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHumanShow
CHEK1 (CHK1)CAMKLCAMK2brgA(5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-aceticHumanShow
CHEK1 (CHK1)CAMKLCAMK2brhAAn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHumanShow
CHEK1 (CHK1)CAMKLCAMK2brhABn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHumanShow
CHEK1 (CHK1)CAMKLCAMK2brmAA3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2brmAB3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2brnA(2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-olHumanShow
CHEK1 (CHK1)CAMKLCAMK2broA(2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diolHumanShow
CHEK1 (CHK1)CAMKLCAMK2c3jAdebromohymenialdisineHumanShow
CHEK1 (CHK1)CAMKLCAMK2c3kA4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenolHumanShow
CHEK1 (CHK1)CAMKLCAMK2c3lA3-(1h-benzimidazol-2-yl)-1h-indazoleHumanShow
CHEK1 (CHK1)CAMKLCAMK2cguA2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acidHumanShow
CHEK1 (CHK1)CAMKLCAMK2cgvA(2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-olHumanShow
CHEK1 (CHK1)CAMKLCAMK2cgwA4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine)HumanShow
CHEK1 (CHK1)CAMKLCAMK2cgxA2-[(6-amino-7h-purin-8-yl)thio]acetamideHumanShow
CHEK1 (CHK1)CAMKLCAMK2e9nA3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamideHumanShow
CHEK1 (CHK1)CAMKLCAMK2e9oA4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHumanShow
CHEK1 (CHK1)CAMKLCAMK2e9pA1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}ureaHumanShow
CHEK1 (CHK1)CAMKLCAMK2e9uA18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2e9vA18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHumanShow
CHEK1 (CHK1)CAMKLCAMK2e9vB18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHumanShow
CHEK1 (CHK1)CAMKLCAMK2gdoA4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2ghgA5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2hogA(5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanolHumanShow
CHEK1 (CHK1)CAMKLCAMK2hxlA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrileHumanShow
CHEK1 (CHK1)CAMKLCAMK2hxqA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2hy0A3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-oneHumanShow
CHEK1 (CHK1)CAMKLCAMK2qhmA(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylateHumanShow
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