PDB-code
Browse kinase entries (page 59 of 282)
First 55 56 57 PreviousLast63 62 61 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CDK9 | CDK | CMGC | 8i0l | A | 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | Show | ![]() | |
![]() | CDK9 | CDK | CMGC | 8k5r | A | (1s,3s)-n3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamine | Human | Show | ![]() | |
![]() | CDKL1 | CDKL | CMGC | 4agu | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | Show | ![]() | |
![]() | CDKL1 | CDKL | CMGC | 4agu | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | Show | ![]() | |
![]() | CDKL1 | CDKL | CMGC | 4agu | C | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | Show | ![]() | |
![]() | CDKL2 | CDKL | CMGC | 4aaa | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | Show | ![]() |
![]() | CDKL2 | CDKL | CMGC | 4aaa | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | Show | ![]() |
![]() | CDKL2 | CDKL | CMGC | 4bbm | A | 4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diol | Human | Show | ![]() | |
![]() | CDKL2 | CDKL | CMGC | 4bbm | B | 4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diol | Human | Show | ![]() | |
![]() | CDKL3 | CDKL | CMGC | 3zdu | A | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | Show | ![]() | |
![]() | CDKL5 | CDKL | CMGC | 4bgq | A | A | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | Show | ![]() |
![]() | CDKL5 | CDKL | CMGC | 4bgq | A | B | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | Show | ![]() |
![]() | CDKL5 | CDKL | CMGC | 8cie | A | 4-[[3,5-bis(fluoranyl)phenyl]carbonylamino]-~{n}-piperidin-4-yl-1~{h}-pyrazole-3-carboxamide | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 1ia8 | A | - | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 1nvq | A | 7-hydroxystaurosporine | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 1nvr | A | staurosporine | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 1nvs | A | rel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dione | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 1zlt | A | (4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-one | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 1zys | A | n-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamide | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2ayp | A | (3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-one | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | A | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | Show | ![]() |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | B | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | Show | ![]() |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2brb | A | 2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanol | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2brg | A | (5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-acetic | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | A | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | Show | ![]() |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | B | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | Show | ![]() |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | A | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | Show | ![]() |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | B | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | Show | ![]() |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2brn | A | (2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-ol | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2bro | A | (2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diol | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2c3j | A | debromohymenialdisine | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2c3k | A | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenol | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2c3l | A | 3-(1h-benzimidazol-2-yl)-1h-indazole | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2cgu | A | 2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acid | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2cgv | A | (2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-ol | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2cgw | A | 4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine) | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2cgx | A | 2-[(6-amino-7h-purin-8-yl)thio]acetamide | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2e9n | A | 3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamide | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2e9o | A | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2e9p | A | 1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}urea | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2e9u | A | 18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-one | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | A | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | B | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2gdo | A | 4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-one | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2ghg | A | 5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2hog | A | (5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanol | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2hxl | A | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrile | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2hxq | A | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-one | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2hy0 | A | 3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-one | Human | Show | ![]() | |
![]() | CHEK1 (CHK1) | CAMKL | CAMK | 2qhm | A | (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylate | Human | Show | ![]() |


