PDB-code
Browse kinase entries (page 61 of 282)
First 57 58 59 PreviousLast65 64 63 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | Show |  |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | A | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | B | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tkh | A | 1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tki | A | n-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3u9n | A | 2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | A | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | B | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | A | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | B | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | A | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | B | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | A | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | B | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | A | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | B | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | A | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | B | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | A | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | B | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | A | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | B | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | A | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | B | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | A | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | B | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | A | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | B | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | A | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | B | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | A | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | B | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | A | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | B | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | A | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | B | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | A | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | B | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | A | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | B | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | A | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | B | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | A | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | B | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | A | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | B | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | A | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | Show | |
