PDB-code
Browse kinase entries (page 62 of 282)
First 58 59 60 PreviousLast66 65 64 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | B | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | Show |  |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | C | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | A | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | B | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | A | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | B | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | A | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | B | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | A | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | B | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | A | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | B | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | A | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | B | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | A | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | B | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | A | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | B | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | A | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | B | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4jik | A | 2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qye | A | 4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyf | A | 4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | A | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | B | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | A | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | B | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvk | A | n-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvl | A | 3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvm | A | 3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5dls | A | 1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | A | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | B | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oor | A | staurosporine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oot | A | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op4 | A | [4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op5 | A | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op7 | A | [4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | A | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | B | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opr | A | 5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5ops | A | 4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opu | A | 6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opv | A | 4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq5 | A | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq6 | A | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | |
