Browse kinase entries (page 67 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CLK1CLKCMGC6yteCB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK1CLKCMGC6ytgAA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK1CLKCMGC6ytgAB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK1CLKCMGC6ytiAAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHumanShow
CLK1CLKCMGC6ytiABmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHumanShow
CLK1CLKCMGC6z4zAA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK1CLKCMGC6z4zAB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK1CLKCMGC6z4zBA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK1CLKCMGC6z4zBB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK1CLKCMGC6z4zCA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK1CLKCMGC6z4zCB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK1CLKCMGC6z50AA11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
CLK1CLKCMGC6z50AB11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
CLK1CLKCMGC6zlnAA4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amineHumanShow
CLK1CLKCMGC6zlnAB4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amineHumanShow
CLK1CLKCMGC7ak3AA~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
CLK1CLKCMGC7ak3AB~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
CLK1CLKCMGC7o9yA4-(1~{h}-indol-3-yl)pyrimidin-2-amineHumanShow
CLK1CLKCMGC7oa0A5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amineHumanShow
CLK1CLKCMGC7opgAA4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenolHumanShow
CLK1CLKCMGC7opgAB4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenolHumanShow
CLK1CLKCMGC8p04A(4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-oneHumanShow
CLK1CLKCMGC8p08A(4~{z})-4-(1,3-benzothiazol-6-ylmethylidene)-2-[[(2~{r})-1-methoxy-4-methyl-pentan-2-yl]amino]-1~{h}-imidazol-5-oneHumanShow
CLK2CLKCMGC3nr9A(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHumanShow
CLK2CLKCMGC3nr9B(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHumanShow
CLK2CLKCMGC3nr9C(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHumanShow
CLK2CLKCMGC5unpAn~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamineHumanShow
CLK2CLKCMGC5unpBn~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamineHumanShow
CLK2CLKCMGC6fyiA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK2CLKCMGC6fykAA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHumanShow
CLK2CLKCMGC6fykAB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHumanShow
CLK2CLKCMGC6fykBA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHumanShow
CLK2CLKCMGC6fykBB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHumanShow
CLK2CLKCMGC6fykCA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHumanShow
CLK2CLKCMGC6fykCB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHumanShow
CLK2CLKCMGC6fylAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK2CLKCMGC6fylAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK2CLKCMGC6kheA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK3CLKCMGC2eu9AA-HumanShow
CLK3CLKCMGC2eu9AB-HumanShow
CLK3CLKCMGC2exeAA-HumanShow
CLK3CLKCMGC2exeAB-HumanShow
CLK3CLKCMGC2wu6AA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHumanShow
CLK3CLKCMGC2wu6AB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHumanShow
CLK3CLKCMGC2wu7AAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHumanShow
CLK3CLKCMGC2wu7ABethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHumanShow
CLK3CLKCMGC3rawAA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
CLK3CLKCMGC3rawAB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
CLK3CLKCMGC3rawBA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
CLK3CLKCMGC3rawBB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
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