PDB-code
Browse kinase entries (page 67 of 282)
First 63 64 65 PreviousLast71 70 69 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CLK1 | CLK | CMGC | 6yte | C | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6ytg | A | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6ytg | A | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6yti | A | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6yti | A | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z4z | A | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z4z | A | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z4z | B | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z4z | B | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z4z | C | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z4z | C | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z50 | A | A | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6z50 | A | B | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6zln | A | A | 4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 6zln | A | B | 4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 7ak3 | A | A | ~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 7ak3 | A | B | ~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 7o9y | A | 4-(1~{h}-indol-3-yl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CLK1 | CLK | CMGC | 7oa0 | A | 5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amine | Human | Show | ![]() | |
![]() | CLK1 | CLK | CMGC | 7opg | A | A | 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 7opg | A | B | 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol | Human | Show | ![]() |
![]() | CLK1 | CLK | CMGC | 8p04 | A | (4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-one | Human | Show | ![]() | |
![]() | CLK1 | CLK | CMGC | 8p08 | A | (4~{z})-4-(1,3-benzothiazol-6-ylmethylidene)-2-[[(2~{r})-1-methoxy-4-methyl-pentan-2-yl]amino]-1~{h}-imidazol-5-one | Human | Show | ![]() | |
![]() | CLK2 | CLK | CMGC | 3nr9 | A | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | Show | ![]() | |
![]() | CLK2 | CLK | CMGC | 3nr9 | B | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | Show | ![]() | |
![]() | CLK2 | CLK | CMGC | 3nr9 | C | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | Show | ![]() | |
![]() | CLK2 | CLK | CMGC | 5unp | A | n~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | CLK2 | CLK | CMGC | 5unp | B | n~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | CLK2 | CLK | CMGC | 6fyi | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | Show | ![]() | |
![]() | CLK2 | CLK | CMGC | 6fyk | A | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6fyk | A | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6fyk | B | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6fyk | B | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6fyk | C | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6fyk | C | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6fyl | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6fyl | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | Show | ![]() |
![]() | CLK2 | CLK | CMGC | 6khe | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | Show | ![]() | |
![]() | CLK3 | CLK | CMGC | 2eu9 | A | A | - | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 2eu9 | A | B | - | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 2exe | A | A | - | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 2exe | A | B | - | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 2wu6 | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 2wu6 | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 2wu7 | A | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 2wu7 | A | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 3raw | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 3raw | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 3raw | B | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | ![]() |
![]() | CLK3 | CLK | CMGC | 3raw | B | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | ![]() |


