Browse kinase entries (page 68 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CLK3CLKCMGC6ft7AA3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHumanShow
CLK3CLKCMGC6ft7AB3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHumanShow
CLK3CLKCMGC6ft7BA3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHumanShow
CLK3CLKCMGC6ft7BB3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHumanShow
CLK3CLKCMGC6fypAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK3CLKCMGC6fypAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK3CLKCMGC6fyrAA6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHumanShow
CLK3CLKCMGC6fyrAB6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHumanShow
CLK3CLKCMGC6khfAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK3CLKCMGC6khfAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK3CLKCMGC6rctAA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHumanShow
CLK3CLKCMGC6rctAB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHumanShow
CLK3CLKCMGC6rctBA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHumanShow
CLK3CLKCMGC6rctBB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHumanShow
CLK3CLKCMGC6ytwAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK3CLKCMGC6ytwAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK3CLKCMGC6ytwBA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK3CLKCMGC6ytwBB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK3CLKCMGC6ytyAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK3CLKCMGC6ytyAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHumanShow
CLK3CLKCMGC6yu1aA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK3CLKCMGC6yu1aB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK3CLKCMGC6yu1cA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK3CLKCMGC6yu1cB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK3CLKCMGC6z2vAA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK3CLKCMGC6z2vAB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHumanShow
CLK3CLKCMGC6z51AAn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide HumanShow
CLK3CLKCMGC6z51ABn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide HumanShow
CLK3CLKCMGC6z52AA11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHumanShow
CLK3CLKCMGC6z52AB11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHumanShow
CLK3CLKCMGC6z52BA11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHumanShow
CLK3CLKCMGC6z52BB11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHumanShow
CLK3CLKCMGC6z53AA6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
CLK3CLKCMGC6z53AB6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
CLK3CLKCMGC6z54AA11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHumanShow
CLK3CLKCMGC6z54AB11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHumanShow
CLK3CLKCMGC6z55AA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK3CLKCMGC6z55AB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK3CLKCMGC6z55AC7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK3CLKCMGC6z55BA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK3CLKCMGC6z55BB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK3CLKCMGC6z55BC7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHumanShow
CLK4CLKCMGC6fyvAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
CLK4CLKCMGC6fyvAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
COQ8A (ADCK3)ABC1Atypical4pedAA-HumanShow
COQ8A (ADCK3)ABC1Atypical4pedAB-HumanShow
COQ8A (ADCK3)ABC1Atypical5i35Aphosphoaminophosphonic acid-adenylate esterHumanShow
COQ8A (ADCK3)ABC1Atypical7udpA4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrileHumanShow
COQ8A (ADCK3)ABC1Atypical7udqA4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrileHumanShow
CSF1R (FMS)PDGFRTK2i0vA6-chloro-3-(3-methylisoxazol-5-yl)-4-phenylquinolin-2(1h)-oneHumanShow
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