Browse kinase entries (page 8 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
ACVR1 (ALK2)STKRTKL5s81AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s82AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s82AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s83AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s83AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s84AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s84AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s84AC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s85AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s85AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s85AC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s86AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s86AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s87AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s87AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s88AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s88AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s89AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s89AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s8aAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s8aAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s8bAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s8bAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s9kAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL5s9kAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL6acrAn-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amineHumanShow
ACVR1 (ALK2)STKRTKL6acrBn-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amineHumanShow
ACVR1 (ALK2)STKRTKL6eixAA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHumanShow
ACVR1 (ALK2)STKRTKL6eixAB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHumanShow
ACVR1 (ALK2)STKRTKL6gi6A5-methyl-6-quinolin-5-yl-3~{h}-quinazolin-4-oneHumanShow
ACVR1 (ALK2)STKRTKL6ginAA3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHumanShow
ACVR1 (ALK2)STKRTKL6ginAB3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHumanShow
ACVR1 (ALK2)STKRTKL6ginBA3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHumanShow
ACVR1 (ALK2)STKRTKL6ginBB3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHumanShow
ACVR1 (ALK2)STKRTKL6gipAA2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-oneHumanShow
ACVR1 (ALK2)STKRTKL6gipAB2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-oneHumanShow
ACVR1 (ALK2)STKRTKL6i1sAA(4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dioneHumanShow
ACVR1 (ALK2)STKRTKL6i1sAB(4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dioneHumanShow
ACVR1 (ALK2)STKRTKL6juxAA4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amineHumanShow
ACVR1 (ALK2)STKRTKL6juxAB4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amineHumanShow
ACVR1 (ALK2)STKRTKL6srhAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL6srhAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL6srhBA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL6srhBB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHumanShow
ACVR1 (ALK2)STKRTKL6szmAA1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHumanShow
ACVR1 (ALK2)STKRTKL6szmAB1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHumanShow
ACVR1 (ALK2)STKRTKL6szmBA1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHumanShow
ACVR1 (ALK2)STKRTKL6szmBB1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHumanShow
ACVR1 (ALK2)STKRTKL6t6dAA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHumanShow
ACVR1 (ALK2)STKRTKL6t6dAB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHumanShow
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