PDB-code
Browse kinase entries (page 71 of 282)
First 67 68 69 PreviousLast75 74 73 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | D | - | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | A | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | B | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | C | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | D | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5ih6 | A | A | 6-(3-bromophenyl)pteridine-2,4,7-triamine | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5ih6 | A | B | 6-(3-bromophenyl)pteridine-2,4,7-triamine | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | A | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | A | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | B | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | B | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | C | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | C | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | D | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | D | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | E | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | E | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | F | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5mqv | F | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | A | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | A | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | B | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | B | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | C | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | C | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | D | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5okt | D | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | A | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | A | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | B | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | B | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | C | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | C | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | D | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 5w4w | D | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f1w | A | A | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f1w | A | B | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f1w | B | A | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f1w | B | B | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | A | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | B | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | C | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | A | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | B | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | C | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6gzm | A | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6gzm | A | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6gzm | B | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6gzm | B | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | Show | ![]() |
![]() | CSNK1D (CK1d) | CK1 | CK1 | 6hmp | A | A | - | Human | Show | ![]() |



